Literature DB >> 21317222

Hemorrhagic complications in a phase II study of sunitinib in patients of nasopharyngeal carcinoma who has previously received high-dose radiation.

E P Hui1, B B Y Ma, A D King, F Mo, S L Chan, M K M Kam, H H Loong, A T Ahuja, B C Y Zee, A T C Chan.   

Abstract

BACKGROUND: We aimed to evaluate the safety and efficacy of single-agent sunitinib in nasopharyngeal carcinoma (NPC).
METHODS: Eligible patients had progressive disease after prior platinum-based chemotherapy. Sunitinib was given as continuous once-daily dosing of 37.5 mg in 4-week cycles until progression.
RESULTS: Thirteen patients were enrolled. Recruitment was stopped after two patients died of hemorrhagic events. All patients had previously received curative radiotherapy (RT) to nasopharynx/neck (including nine patients who had chemoradiotherapy). Patients received a median of three cycles of sunitinib. One patient was still on sunitinib with stable disease after 24 cycles. Hemorrhagic events occurred in nine patients (64%), including epistaxis in six, hemoptyses in three and hematemesis in two patients. Prior RT to thorax was significantly associated with hemoptyses (P = 0.03). Two patients with local tumor invasion into the carotid sheath developed fatal epistaxis/hematemesis within the first cycle of sunitinib, likely due to internal carotid blowout after tumor shrinkage.
CONCLUSIONS: Sunitinib demonstrated modest clinical activity in heavily pretreated NPC patients. However, the high incidence of hemorrhage from the upper aerodigestive tract in NPC patients who received prior high-dose RT to the region is of concern. Direct vascular invasion by tumors appeared to increase the risk of serious bleeding.

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Year:  2011        PMID: 21317222     DOI: 10.1093/annonc/mdq629

Source DB:  PubMed          Journal:  Ann Oncol        ISSN: 0923-7534            Impact factor:   32.976


  33 in total

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2.  Lenvatinib as a novel treatment for anaplastic thyroid cancer: A retrospective study.

Authors:  Hiroyuki Iwasaki; Haruhiko Yamazaki; Hirotaka Takasaki; Nobuyasu Suganuma; Hirotaka Nakayama; Soji Toda; Katsuhiko Masudo
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Review 3.  Combining targeted agents with modern radiotherapy in soft tissue sarcomas.

Authors:  Philip Wong; Peter Houghton; David G Kirsch; Steven E Finkelstein; Arta M Monjazeb; Meng Xu-Welliver; Adam P Dicker; Mansoor Ahmed; Bhadrasain Vikram; Beverly A Teicher; C Norman Coleman; Mitchell Machtay; Walter J Curran; Dian Wang
Journal:  J Natl Cancer Inst       Date:  2014-10-18       Impact factor: 13.506

4.  Optimizing the Sunitinib for cardio-toxicity and thyro-toxicity by scaffold hopping approach.

Authors:  Bhagyashri Chaudhari; Harun Patel; Snehal Thakar; Iqrar Ahmad; Deepali Bansode
Journal:  In Silico Pharmacol       Date:  2022-07-02

Review 5.  Nasopharyngeal carcinoma: an evolving paradigm.

Authors:  Kenneth C W Wong; Edwin P Hui; Kwok-Wai Lo; Wai Kei Jacky Lam; David Johnson; Lili Li; Qian Tao; Kwan Chee Allen Chan; Ka-Fai To; Ann D King; Brigette B Y Ma; Anthony T C Chan
Journal:  Nat Rev Clin Oncol       Date:  2021-06-30       Impact factor: 66.675

6.  Multicenter phase II study of the AKT inhibitor MK-2206 in recurrent or metastatic nasopharyngeal carcinoma from patients in the mayo phase II consortium and the cancer therapeutics research group (MC1079).

Authors:  B B Y Ma; B C Goh; W T Lim; E P Hui; E H Tan; G de Lima Lopes; K W Lo; L Li; H Loong; N R Foster; C Erlichman; A D King; M K M Kam; S F Leung; K C Chan; A T C Chan
Journal:  Invest New Drugs       Date:  2015-06-19       Impact factor: 3.651

7.  Treatment of nasopharyngeal carcinoma cells with the histone-deacetylase inhibitor abexinostat: cooperative effects with cis-platin and radiotherapy on patient-derived xenografts.

Authors:  Mélanie Gressette; Benjamin Vérillaud; Anne-Sophie Jimenez-Pailhès; Hélène Lelièvre; Kwok-Wai Lo; François-Régis Ferrand; Charles-Henry Gattolliat; Anne Jacquet-Bescond; Laurence Kraus-Berthier; Stéphane Depil; Pierre Busson
Journal:  PLoS One       Date:  2014-03-11       Impact factor: 3.240

8.  Fatal bleeding in a nasopharyngeal carcinoma patient after concurrent chemoradiation plus cetuximab: a case report.

Authors:  Lingyan Zheng; Senxiang Yan; Danfang Yan; Jingsong Yang; Yixiang Wang
Journal:  Onco Targets Ther       Date:  2013-06-13       Impact factor: 4.147

Review 9.  Emerging treatment options for nasopharyngeal carcinoma.

Authors:  Lu Zhang; Qiu-Yan Chen; Huai Liu; Lin-Quan Tang; Hai-Qiang Mai
Journal:  Drug Des Devel Ther       Date:  2013-02-01       Impact factor: 4.162

10.  Met tyrosine kinase inhibitor, PF-2341066, suppresses growth and invasion of nasopharyngeal carcinoma.

Authors:  Yuanyuan Zhao; Jing Zhang; Ying Tian; Cong Xue; Zhihuang Hu; Li Zhang
Journal:  Drug Des Devel Ther       Date:  2015-08-26       Impact factor: 4.162

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