Literature DB >> 21314107

Synthesis of α-carbolines via Pd-catalyzed amidation and Vilsmeier-Haack reaction of 3-acetyl-2-chloroindoles.

Arepalli Sateesh Kumar1, Rajagopal Nagarajan.   

Abstract

A new class of α-carboline derivatives has been synthesized by Pd(2)(dba)(3)/BINAP catalyzed amidation of 3-acetyl-2-chloroindoles followed by a Vilsmeier-Haack reaction and is reported.

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Year:  2011        PMID： 21314107     DOI： 10.1021/ol2000827

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  6 in total

1.  A simple and facile synthesis of tricyclic-fused pyrimido[4,5-b]indol-2-amines.

Authors:  Wentao Gao; Dongfang Wang; Yang Li
Journal:  Mol Divers       Date:  2017-06-19       Impact factor: 2.943

2.  Rh(II)2-catalyzed synthesis of α-, β-, or δ-carbolines from aryl azides.

Authors:  Ashley L Pumphrey; Huijun Dong; Tom G Driver
Journal:  Angew Chem Int Ed Engl       Date:  2012-04-26       Impact factor: 15.336

Review 3.  Applications of Palladium-Catalyzed C-N Cross-Coupling Reactions.

Authors:  Paula Ruiz-Castillo; Stephen L Buchwald
Journal:  Chem Rev       Date:  2016-09-30       Impact factor: 60.622

4.  An intramolecular inverse electron demand Diels-Alder approach to annulated α-carbolines.

Authors:  Zhiyuan Ma; Feng Ni; Grace H C Woo; Sie-Mun Lo; Philip M Roveto; Scott E Schaus; John K Snyder
Journal:  Beilstein J Org Chem       Date:  2012-06-06       Impact factor: 2.883

5.  Nigritanine as a New Potential Antimicrobial Alkaloid for the Treatment of Staphylococcus aureus-Induced Infections.

Authors:  Bruno Casciaro; Andrea Calcaterra; Floriana Cappiello; Mattia Mori; Maria Rosa Loffredo; Francesca Ghirga; Maria Luisa Mangoni; Bruno Botta; Deborah Quaglio
Journal:  Toxins (Basel)       Date:  2019-09-01       Impact factor: 4.546

6.  A new route to α-carbolines based on 6π-electrocyclization of indole-3-alkenyl oximes.

Authors:  Sophie J Markey; William Lewis; Christopher J Moody
Journal:  Org Lett       Date:  2013-11-26       Impact factor: 6.005
  6 in total

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