Literature DB >> 21190067

Influence of acylation on the adsorption of insulin to hydrophobic surfaces.

Charlotte Pinholt1, Susanne Hostrup, Jens Thostrup Bukrinsky, Sven Frokjaer, Lene Jorgensen.   

Abstract

PURPOSE: To study the effect of acylation on the adsorption of insulin to hydrophobic polystyrene beads.
METHODS: Adsorption isotherms for adsorption of insulin and acylated insulin to hydrophobic polystyrene beads were established, and the adsorption of the two proteins was compared further with isothermal titration calorimetry. In addition, the secondary structure and the association behavior of the two proteins were studied with circular dichroism.
RESULTS: Insulin and acylated insulin adsorbed with high affinity to the hydrophobic polystyrene beads. More acylated insulin molecules than insulin molecules adsorbed per unit surface area from solutions containing monomer-dimer mixtures of acylated insulin and insulin, respectively. In contrast, no difference was observed in the number of insulin and acylated insulin molecules adsorbing per unit surface area, when adsorption occurred from solutions containing monomer-dimer-hexamer mixtures.
CONCLUSION: The influence of acylation on the adsorption behavior of insulin depends on the association degree of insulin, possibly due to a greater difference in hydrophobicity between monomeric insulin and acylated insulin than between the hexameric forms of these two proteins.

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Year:  2010        PMID: 21190067     DOI: 10.1007/s11095-010-0349-6

Source DB:  PubMed          Journal:  Pharm Res        ISSN: 0724-8741            Impact factor:   4.200


  27 in total

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Authors:  P Krüger; G Gilge; Y Cabuk; A Wollmer
Journal:  Biol Chem Hoppe Seyler       Date:  1990-08

2.  Reversible lipidization for the oral delivery of leu-enkephalin.

Authors:  Jeffrey Wang; Derk J Hogenkamp; Minhtam Tran; Wen-Yen Li; Ryan F Yoshimura; Timothy B C Johnstone; Wei-Chiang Shen; Kelvin W Gee
Journal:  J Drug Target       Date:  2006-04       Impact factor: 5.121

3.  Adsorption of human insulin and AspB28 insulin on a PTFE-like surface.

Authors:  S H Mollmann; J T Bukrinsky; S Frokjaer; U Elofsson
Journal:  J Colloid Interface Sci       Date:  2005-06-01       Impact factor: 8.128

4.  Preparation, purification, and characterization of a reversibly lipidized desmopressin with potentiated anti-diuretic activity.

Authors:  J Wang; D Shen; W C Shen
Journal:  Pharm Res       Date:  1999-11       Impact factor: 4.200

5.  Reversible lipidization prolongs the pharmacological effect, plasma duration, and liver retention of octreotide.

Authors:  Liyun Yuan; Jeff Wang; Wei-Chiang Shen
Journal:  Pharm Res       Date:  2005-02       Impact factor: 4.200

6.  Adsorption Kinetics, Conformation, and Mobility of the Growth Hormone and Lysozyme on Solid Surfaces, Studied with TIRF

Authors: 
Journal:  J Colloid Interface Sci       Date:  1997-06-01       Impact factor: 8.128

7.  Soluble, fatty acid acylated insulins bind to albumin and show protracted action in pigs.

Authors:  J Markussen; S Havelund; P Kurtzhals; A S Andersen; J Halstrøm; E Hasselager; U D Larsen; U Ribel; L Schäffer; K Vad; I Jonassen
Journal:  Diabetologia       Date:  1996-03       Impact factor: 10.122

8.  Partially folded intermediates in insulin fibrillation.

Authors:  Atta Ahmad; Ian S Millett; Sebastian Doniach; Vladimir N Uversky; Anthony L Fink
Journal:  Biochemistry       Date:  2003-10-07       Impact factor: 3.162

9.  The mechanism of protraction of insulin detemir, a long-acting, acylated analog of human insulin.

Authors:  Svend Havelund; Anne Plum; Ulla Ribel; Ib Jonassen; Aage Vølund; Jan Markussen; Peter Kurtzhals
Journal:  Pharm Res       Date:  2004-08       Impact factor: 4.200

10.  Solution structure and biological activity of recombinant salmon calcitonin S-sulfonated analog.

Authors:  Yuefeng Wang; Hong Dou; Chunyang Cao; Naixia Zhang; Jingbiao Ma; Jifang Mao; Houming Wu
Journal:  Biochem Biophys Res Commun       Date:  2003-06-27       Impact factor: 3.575

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