Literature DB >> 2116800

Lysis of trypanosomes by peptidyl fluoromethyl ketones.

F Ashall1, H Angliker, E Shaw.   

Abstract

Peptidyl fluoromethyl ketones, improved reagents for inactivating cysteinyl and serine proteinases, have provided unexpected results when applied to intact trypanosomes. A lethal effect was observed but limited to the infectious phase of the parasitic growth cycle. Since the inhibitors are known only to act on proteases, the result implies the existence of a protease of critical importance during the infectious phase. A labelled inhibitor, Cbz-Ala-[3H]Phe-CH2F, indicated that the killing effect correlated with the labelling of a 68 kd protein in the trypomastigotes which we deduce is an essential protease.

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Year:  1990        PMID: 2116800     DOI: 10.1016/0006-291x(90)92179-4

Source DB:  PubMed          Journal:  Biochem Biophys Res Commun        ISSN: 0006-291X            Impact factor:   3.575


  5 in total

1.  Discovery of trypanocidal thiosemicarbazone inhibitors of rhodesain and TbcatB.

Authors:  Jeremy P Mallari; Anang Shelat; Aaron Kosinski; Conor R Caffrey; Michele Connelly; Fangyi Zhu; James H McKerrow; R Kiplin Guy
Journal:  Bioorg Med Chem Lett       Date:  2008-04-08       Impact factor: 2.823

2.  Trypanosomatid cysteine protease activity may be enhanced by a kininogen-like moiety from host serum.

Authors:  J D Lonsdale-Eccles; G W Mpimbaza; Z R Nkhungulu; J Olobo; L Smith; O M Tosomba; D J Grab
Journal:  Biochem J       Date:  1995-01-15       Impact factor: 3.857

3.  The cysteine proteinase inhibitor Z-Phe-Ala-CHN2 alters cell morphology and cell division activity of Trypanosoma brucei bloodstream forms in vivo.

Authors:  Stefan Scory; York-Dieter Stierhof; Conor R Caffrey; Dietmar Steverding
Journal:  Kinetoplastid Biol Dis       Date:  2007-02-28

4.  Novel scaffolds for inhibition of Cruzipain identified from high-throughput screening of anti-kinetoplastid chemical boxes.

Authors:  Emir Salas-Sarduy; Lionel Urán Landaburu; Joel Karpiak; Kevin P Madauss; Juan José Cazzulo; Fernán Agüero; Vanina Eder Alvarez
Journal:  Sci Rep       Date:  2017-09-21       Impact factor: 4.379

5.  Cysteine protease inhibitors cure an experimental Trypanosoma cruzi infection.

Authors:  J C Engel; P S Doyle; I Hsieh; J H McKerrow
Journal:  J Exp Med       Date:  1998-08-17       Impact factor: 14.307

  5 in total

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