Literature DB >> 21118280

The 12-month safety profile of dexlansoprazole, a proton pump inhibitor with a dual delayed release formulation, in patients with gastro-oesophageal reflux disease.

A H Dabholkar1, C Han, M M Paris, M C Perez, S N Atkinson, D A Peura.   

Abstract

BACKGROUND: Dexlansoprazole MR is a Dual Delayed Release formulation of dexlansoprazole, an enantiomer of lansoprazole, designed to extend the duration of acid suppression. AIM: To assess the 12-month safety of dexlansoprazole MR in patients with symptomatic gastro-oesophageal reflux disease (GERD).
METHODS: In this randomised open-label study, patients received dexlansoprazole MR 60 or 90 mg once-daily for 12 months. Safety was evaluated at months 1, 3, 6, 9 and 12/final visit through physical examinations, laboratory evaluations, endoscopies, gastric biopsies, fasting serum gastrin values and adverse events (AEs).
RESULTS: Of 591 patients receiving dexlansoprazole MR 60 and 90 mg, 71% and 65%, respectively, experienced ≥1 treatment-emergent AE; the most frequent AE was upper respiratory infection (14% and 13% in the 60- and 90-mg groups). Thirty patients experienced ≥1 serious AE; a majority of serious AEs were unrelated to study drug. No clinically meaningful change in any clinical laboratory parameters was noted. As expected, serum gastrin values rose with dexlansoprazole therapy; increases were not dose related. No clinically concerning trends were identified in gastric pathology results; no endocrine cell hyperplasia, adenocarcinoma, or lymphoma were observed.
CONCLUSIONS: Twelve-month treatment with dexlansoprazole MR 60 and 90 mg was well tolerated by GERD patients in this study (Clinicaltrials.gov identifier NCT00255190).
© 2010 Blackwell Publishing Ltd.

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Year:  2010        PMID: 21118280     DOI: 10.1111/j.1365-2036.2010.04519.x

Source DB:  PubMed          Journal:  Aliment Pharmacol Ther        ISSN: 0269-2813            Impact factor:   8.171


  5 in total

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Authors:  Taline A Boghossian; Farah Joy Rashid; Wade Thompson; Vivian Welch; Paul Moayyedi; Carlos Rojas-Fernandez; Kevin Pottie; Barbara Farrell
Journal:  Cochrane Database Syst Rev       Date:  2017-03-16

Review 2.  Dexlansoprazole - a new-generation proton pump inhibitor.

Authors:  Barbara Skrzydło-Radomańska; Piotr Radwan
Journal:  Prz Gastroenterol       Date:  2015-12-16

Review 3.  Proton pump inhibitors for the treatment of patients with erosive esophagitis and gastroesophageal reflux disease: current evidence and safety of dexlansoprazole.

Authors:  Joseph Mermelstein; Alanna Chait Mermelstein; Maxwell M Chait
Journal:  Clin Exp Gastroenterol       Date:  2016-07-13

4.  Effectiveness and Tolerability of Different Recommended Doses of PPIs and H2RAs in GERD: Network Meta-Analysis and GRADE system.

Authors:  Chao Zhang; Joey S W Kwong; Rui-Xia Yuan; Hao Chen; Chang Xu; Yi-Pin Wang; Gong-Li Yang; Jin-Zhu Yan; Le Peng; Xian-Tao Zeng; Hong Weng; Jie Luo; Yu-Ming Niu
Journal:  Sci Rep       Date:  2017-01-19       Impact factor: 4.379

5.  Bioavailability of a dexlansoprazole delayed-release orally disintegrating tablet: effects of food and mode of administration.

Authors:  Michael Kukulka; Sai Nudurupati; Maria Claudia Perez
Journal:  Clin Exp Gastroenterol       Date:  2017-02-17
  5 in total

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