Literature DB >> 21094564

Synthesis and antimycobacterial activity of a series of ferrocenyl derivatives.

Gabin Mwande Maguene1, Jouda Jakhlal, Melissa Ladyman, Aurélie Vallin, Dimby Andrianina Ralambomanana, Till Bousquet, Jeanne Maugein, Jacques Lebibi, Lydie Pélinski.   

Abstract

In this work we reported the synthesis and evaluation of Mycobacterium tuberculosis activities in vitro of a series of twenty five ferrocenyl derivatives: ferrocenyl amides derived from nicotinamide and pyrazinamide, ferrocenyl pyridinyl, quinolyl and acridinylhydrazones. In particular ferrocenyl acylhydrazones 7 and 8 and ferrocenylquinoxaline amide 57 showed interesting antimycobacterial activities.
Copyright © 2010. Published by Elsevier Masson SAS.

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Year:  2010        PMID: 21094564     DOI: 10.1016/j.ejmech.2010.10.004

Source DB:  PubMed          Journal:  Eur J Med Chem        ISSN: 0223-5234            Impact factor:   6.514


  3 in total

1.  Crystal structures of two hydrazide derivatives of mefenamic acid, 3-(2,3-di-methyl-anilino)-N'-[(E)-(furan-2-yl)methyl-idene]benzohydrazide and N'-[(E)-benzyl-idene]-2-(2,3-di-methyl-anilino)benzo-hydrazide.

Authors:  Shaaban K Mohamed; Joel T Mague; Mehmet Akkurt; Mustafa R Albayati; Sahar M I Elgarhy; Elham A Al-Taifi
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2021-02-12

2.  Enantiomeric-Enriched Ferrocenes: Synthesis, Chiral Resolution, and Mathematic Evaluation of CD-chiral Selector Energies with Ferrocene-Conjugates.

Authors:  Lubov V Snegur; Yurii A Borisov; Yuliya V Kuzmenko; Vadim A Davankov; Mikhail M Ilyin; Mikhail M Ilyin; Dmitry E Arhipov; Alexander A Korlyukov; Sergey S Kiselev; Alexander A Simenel
Journal:  Molecules       Date:  2017-08-25       Impact factor: 4.411

3.  New sulfonamides containing organometallic-acylhydrazones: synthesis, characterisation and biological evaluation as inhibitors of human carbonic anhydrases.

Authors:  Yosselin Huentupil; Luis Peña; Néstor Novoa; Emanuela Berrino; Rodrigo Arancibia; Claudiu T Supuran
Journal:  J Enzyme Inhib Med Chem       Date:  2019-12       Impact factor: 5.051

  3 in total

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