Literature DB >> 20963222

A borylative cyclisation towards indole boronic esters.

Jianhui Huang1, Simon J F Macdonald, Joseph P A Harrity.   

Abstract

2-Alkynylaniline borylative cyclisations provide a direct means to access indole 3-boronic esters from simple precursors. The Pd-catalysed cyclisation can be merged with cross-coupling processes in the same reaction vessel, moreover, the products can be exploited in C-N bond forming reactions.

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Year:  2010        PMID: 20963222     DOI: 10.1039/c0cc03577g

Source DB:  PubMed          Journal:  Chem Commun (Camb)        ISSN: 1359-7345            Impact factor:   6.222


  4 in total

1.  BCl3 -Induced Annulative Oxo- and Thioboration for the Formation of C3-Borylated Benzofurans and Benzothiophenes.

Authors:  Andrew J Warner; Anna Churn; John S McGough; Michael J Ingleson
Journal:  Angew Chem Int Ed Engl       Date:  2016-11-29       Impact factor: 15.336

Review 2.  Indolylboronic Acids: Preparation and Applications.

Authors:  Marek Čubiňák; Tereza Edlová; Peter Polák; Tomáš Tobrman
Journal:  Molecules       Date:  2019-09-28       Impact factor: 4.411

3.  Aminoboration: Addition of B-N σ Bonds across C-C π Bonds.

Authors:  Eugene Chong; Suzanne A Blum
Journal:  J Am Chem Soc       Date:  2015-08-10       Impact factor: 15.419

4.  Formation of C(sp(2))-boronate esters by borylative cyclization of alkynes using BCl3.

Authors:  Andrew J Warner; James R Lawson; Valerio Fasano; Michael J Ingleson
Journal:  Angew Chem Int Ed Engl       Date:  2015-07-31       Impact factor: 15.336

  4 in total

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