Literature DB >> 20938715

A phase II open-label trial of bortezomib in patients with multiple myeloma who have undergone an autologous peripheral blood stem cell transplant and failed to achieve a complete response.

Robert M Rifkin1, Andrew Greenspan, John F Schwerkoske, Romeo A Mandanas, Joe J Stephenson, George T Kannarkat, Feng Zhan, Kristi A Boehm, Lina Asmar, Roy Beveridge.   

Abstract

BACKGROUND: A majority of multiple myeloma (MM) patients fail to achieve complete response (CR) to peripheral blood stem cell transplantation (PBSCT); effective options following autologous transplantation are needed. Bortezomib (B) is active against MM. This study was conducted to determine the feasibility, safety, tolerability, and efficacy of B following high-dose melphalan therapy and PBSCT. Methods Fifty patients enrolled (48 evaluable) and 49 were treated (safety population). TREATMENT: 4 cycles B 1.3 mg/m(2) Days 1, 4, 8, and 11/21-days; 4 additional cycles were permitted for stable or responding patients. Results Median age was 55 years (range, 38-73), 68% male, 64% ECOG PS = 0, 44% Durie-Salmon Stage IIIA prior to induction, 42% had symptomatic IgG MM; 74% had prior single transplant (26% tandem). Responses post-transplant: 70% PRs, 18% MRs. A median of 4 cycles (range, 2-8) of B were administered. Responses: CR 8%, uCR 2%, PR 23%, uPR 19%, MR 10%, and no change 35%; median time-to-treatment failure (TTF) was 6.2 months (range, 1.0-19.4). Three deaths occurred (n = 1 sepsis, n = 2 disease progression). Grade 3-4 treatment-related toxicities included: thrombocytopenia, neuropathy (14%, each); asthenia, neutropenia (10%, each); and nausea (4%). Twelve patients (24%) discontinued treatment due to toxicity and 30 patients (60%) completed the study; 20 patients started new treatment (median 5.8 months [range, 1.5-20.3]).
CONCLUSIONS: The study closed early due to widespread availability of B, and the lack of B-naïve patients. Bortezomib monotherapy after melphalan and autologous PBSCT was feasible, safe and well-tolerated (toxicities were manageable), but failed to produce the hypothesized response rates.

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Year:  2010        PMID: 20938715     DOI: 10.1007/s10637-010-9556-6

Source DB:  PubMed          Journal:  Invest New Drugs        ISSN: 0167-6997            Impact factor:   3.850


  7 in total

1.  High-dose melphalan with autotransplantation for refractory multiple myeloma: results of a Southwest Oncology Group phase II trial.

Authors:  D H Vesole; J J Crowley; R Catchatourian; P J Stiff; D B Johnson; J Cromer; S E Salmon; B Barlogie
Journal:  J Clin Oncol       Date:  1999-07       Impact factor: 44.544

2.  Efficacy and safety of bortezomib in patients with renal impairment: results from the APEX phase 3 study.

Authors:  J F San-Miguel; P G Richardson; P Sonneveld; M W Schuster; D Irwin; E A Stadtmauer; T Facon; J-L Harousseau; D Ben-Yehuda; S Lonial; H Goldschmidt; D Reece; J Bladé; M Boccadoro; J D Cavenagh; R Neuwirth; A L Boral; D-L Esseltine; K C Anderson
Journal:  Leukemia       Date:  2008-01-17       Impact factor: 11.528

3.  Incorporating bortezomib into upfront treatment for multiple myeloma: early results of total therapy 3.

Authors:  Bart Barlogie; Elias Anaissie; Frits van Rhee; Jeffrey Haessler; Klaus Hollmig; Mauricio Pineda-Roman; Michele Cottler-Fox; Abid Mohiuddin; Yazan Alsayed; Guido Tricot; Vanessa Bolejack; Maurizio Zangari; Joshua Epstein; Nathan Petty; Douglas Steward; Bonnie Jenkins; Jennifer Gurley; Ellen Sullivan; John Crowley; John D Shaughnessy
Journal:  Br J Haematol       Date:  2007-07       Impact factor: 6.998

Review 4.  The role of stem cell transplantation in multiple myeloma.

Authors:  Jean-Luc Harousseau; Michel Attal
Journal:  Blood Rev       Date:  2002-12       Impact factor: 8.250

5.  A phase 2 study of bortezomib in relapsed, refractory myeloma.

Authors:  Paul G Richardson; Bart Barlogie; James Berenson; Seema Singhal; Sundar Jagannath; David Irwin; S Vincent Rajkumar; Gordan Srkalovic; Melissa Alsina; Raymond Alexanian; David Siegel; Robert Z Orlowski; David Kuter; Steven A Limentani; Stephanie Lee; Teru Hideshima; Dixie-Lee Esseltine; Michael Kauffman; Julian Adams; David P Schenkein; Kenneth C Anderson
Journal:  N Engl J Med       Date:  2003-06-26       Impact factor: 91.245

6.  Criteria for evaluating disease response and progression in patients with multiple myeloma treated by high-dose therapy and haemopoietic stem cell transplantation. Myeloma Subcommittee of the EBMT. European Group for Blood and Marrow Transplant.

Authors:  J Bladé; D Samson; D Reece; J Apperley; B Björkstrand; G Gahrton; M Gertz; S Giralt; S Jagannath; D Vesole
Journal:  Br J Haematol       Date:  1998-09       Impact factor: 6.998

7.  Bortezomib administered pre-auto-SCT and as maintenance therapy post transplant for multiple myeloma: a single institution phase II study.

Authors:  G L Uy; S D Goyal; N M Fisher; A Y Oza; M H Tomasson; K Stockerl-Goldstein; J F DiPersio; R Vij
Journal:  Bone Marrow Transplant       Date:  2008-11-24       Impact factor: 5.483

  7 in total
  2 in total

1.  Meta-analysis of incidence and risk of peripheral neuropathy associated with intravenous bortezomib.

Authors:  Ling Peng; Xianghua Ye; Yun Zhou; Junyan Zhang; Qiong Zhao
Journal:  Support Care Cancer       Date:  2015-02-13       Impact factor: 3.603

2.  Infliction of proteotoxic stresses by impairment of the unfolded protein response or proteasomal inhibition as a therapeutic strategy for mast cell leukemia.

Authors:  Thomas Wilhelm; Fabian Bick; Kerstin Peters; Vrinda Mohta; Boaz Tirosh; John B Patterson; Behzad Kharabi-Masouleh; Michael Huber
Journal:  Oncotarget       Date:  2017-12-17
  2 in total

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