Literature DB >> 20924097

Improvement in left ventricular systolic and diastolic performance during ranolazine treatment in patients with stable angina.

Vincent M Figueredo1, Gregg S Pressman, Abel Romero-Corral, Elmer Murdock, Pat Holderbach, D Lynn Morris.   

Abstract

PURPOSE: Ranolazine is a novel antianginal medication that acts by ameliorating disturbed sodium and calcium homeostasis. By preventing myocyte sodium and calcium overload, ranolazine also have potential beneficial effects on myocardial function. Experimental models support this concept, as do 2 small studies in human participants receiving ranolazine intravenously. We evaluated changes in parameters of left ventricular function in stable angina patients treated with oral ranolazine.
METHODS: Twenty-two participants were enrolled with Doppler echocardiography performed at baseline and a mean of 2 months after initiation of treatment.
RESULTS: Global left ventricular function, as assessed by the myocardial performance index, was significantly improved on drug therapy (P < .0001). This was due to improvement in both diastolic and systolic parameters. Of 21 patients, 17 reported less angina and 8 patients reported an increase in activity level.
CONCLUSIONS: We report improved parameters of left ventricular function in response to ranolazine as used in the clinical setting.

Entities:  

Mesh:

Substances:

Year:  2010        PMID: 20924097     DOI: 10.1177/1074248410382105

Source DB:  PubMed          Journal:  J Cardiovasc Pharmacol Ther        ISSN: 1074-2484            Impact factor:   2.457


  16 in total

1.  CrossTalk proposal: The late sodium current is an important player in the development of diastolic heart failure (heart failure with a preserved ejection fraction).

Authors:  Marc Pourrier; Sarah Williams; Donald McAfee; Luiz Belardinelli; David Fedida
Journal:  J Physiol       Date:  2014-02-01       Impact factor: 5.182

2.  Rebuttal from Zoltan Papp, Attila Borbely and Walter J. Paulus.

Authors:  Zoltán Papp; Attila Borbély; Walter J Paulus
Journal:  J Physiol       Date:  2014-02-01       Impact factor: 5.182

Review 3.  Left ventricular diastolic dysfunction in women with nonobstructive ischemic heart disease: insights from magnetic resonance imaging and spectroscopy.

Authors:  Michael D Nelson
Journal:  Am J Physiol Regul Integr Comp Physiol       Date:  2017-08-09       Impact factor: 3.619

Review 4.  Ranolazine: a review of its use as add-on therapy in patients with chronic stable angina pectoris.

Authors:  Gillian M Keating
Journal:  Drugs       Date:  2013-01       Impact factor: 9.546

5.  Ranolazine prevents pressure overload-induced cardiac hypertrophy and heart failure by restoring aberrant Na+ and Ca2+ handling.

Authors:  Jiali Nie; Quanlu Duan; Mengying He; Xianqing Li; Bei Wang; Chi Zhou; Lujin Wu; Zheng Wen; Chen Chen; Dao Wu Wang; Katherina M Alsina; Xander H T Wehrens; Dao Wen Wang; Li Ni
Journal:  J Cell Physiol       Date:  2018-11-29       Impact factor: 6.384

Review 6.  Anti-anginal and anti-ischemic effects of late sodium current inhibition.

Authors:  Neil J Wimmer; Peter H Stone
Journal:  Cardiovasc Drugs Ther       Date:  2013-02       Impact factor: 3.727

7.  Effect of ranolazine on left ventricular dyssynchrony in patients with coronary artery disease.

Authors:  Rajesh Venkataraman; Ji Chen; Ernest V Garcia; Luiz Belardinelli; Fadi G Hage; Jaekyeong Heo; Ami E Iskandrian
Journal:  Am J Cardiol       Date:  2012-08-10       Impact factor: 2.778

Review 8.  New strategies for heart failure with preserved ejection fraction: the importance of targeted therapies for heart failure phenotypes.

Authors:  Michele Senni; Walter J Paulus; Antonello Gavazzi; Alan G Fraser; Javier Díez; Scott D Solomon; Otto A Smiseth; Marco Guazzi; Carolyn S P Lam; Aldo P Maggioni; Carsten Tschöpe; Marco Metra; Scott L Hummel; Frank Edelmann; Giuseppe Ambrosio; Andrew J Stewart Coats; Gerasimos S Filippatos; Mihai Gheorghiade; Stefan D Anker; Daniel Levy; Marc A Pfeffer; Wendy Gattis Stough; Burkert M Pieske
Journal:  Eur Heart J       Date:  2014-08-07       Impact factor: 29.983

9.  Effects of ranolazine in a model of doxorubicin-induced left ventricle diastolic dysfunction.

Authors:  Donato Cappetta; Grazia Esposito; Raffaele Coppini; Elena Piegari; Rosa Russo; Loreta Pia Ciuffreda; Alessia Rivellino; Lorenzo Santini; Concetta Rafaniello; Cristina Scavone; Francesco Rossi; Liberato Berrino; Konrad Urbanek; Antonella De Angelis
Journal:  Br J Pharmacol       Date:  2017-05-16       Impact factor: 8.739

Review 10.  New treatment options for late Na current, arrhythmias, and diastolic dysfunction.

Authors:  Lars S Maier
Journal:  Curr Heart Fail Rep       Date:  2012-09
View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.