Literature DB >> 20871394

Neurokinin-1 and novel serotonin antagonists for postoperative and postdischarge nausea and vomiting.

Elizabeth George1, Cyrill Hornuss, Christian C Apfel.   

Abstract

PURPOSE OF REVIEW: This review will address novel options for the prevention and treatment of postoperative and postdischarge nausea and vomiting (PONV and PDNV) after ambulatory anesthesia. In particular, this paper will review the characteristics of neurokinin-1 receptor antagonists (NK1-RAs) and the new serotonin receptor antagonist (5HT3-RA) palonosetron. Finally, we will discuss strategies for prophylaxis and treatment of PONV and PDNV that address the unique concerns in ambulatory surgery patients. RECENT
FINDINGS: First, although PONV has previously been recognized to be a problem for inpatients, new research suggests that the incidence of PDNV after ambulatory surgery may be as high as 35%. Second, NK1-RAs, including aprepitant, the first approved member of this family, are significantly more efficacious than any other antiemetic for the prevention of vomiting. They are however not more effective than other interventions for the control of nausea. Third, the next generation of 5HT3-RAs, such as palonosetron, does not affect the QT interval and has a half-life of 40 h that should be advantageous for the prevention of PDNV.
SUMMARY: Because of the high incidence of PDNV, a predictive model for PDNV would be helpful to determine appropriate antiemetic interventions for each individual patient. Drugs that may be particularly favorable are the novel NK1-RA aprepitant and the next generation 5HT3-RA palonosetron.

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Year:  2010        PMID: 20871394     DOI: 10.1097/ACO.0b013e32833f9f7b

Source DB:  PubMed          Journal:  Curr Opin Anaesthesiol        ISSN: 0952-7907            Impact factor:   2.706


  6 in total

Review 1.  Update on the management of postoperative nausea and vomiting.

Authors:  Anthony L Kovac
Journal:  Drugs       Date:  2013-09       Impact factor: 9.546

2.  Postdischarge Nausea and Vomiting Remains Frequent After Le Fort I Osteotomy Despite Implementation of a Multimodal Antiemetic Protocol Effective in Reducing Postoperative Nausea and Vomiting.

Authors:  Carolyn Dicus Brookes; Timothy A Turvey; Ceib Phillips; Vincent Kopp; Jay A Anderson
Journal:  J Oral Maxillofac Surg       Date:  2015-01-29       Impact factor: 1.895

Review 3.  Neurokinin-1 inhibitors in the prevention of nausea and vomiting from highly emetogenic chemotherapy: a network meta-analysis.

Authors:  Omar Abdel-Rahman
Journal:  Ther Adv Med Oncol       Date:  2016-06-29       Impact factor: 8.168

4.  Multimodal protocol reduces postoperative nausea and vomiting in patients undergoing Le Fort I osteotomy.

Authors:  Carolyn Dicus Brookes; John Berry; Josiah Rich; Brent A Golden; Timothy A Turvey; George Blakey; Vincent Kopp; Ceib Phillips; Jay Anderson
Journal:  J Oral Maxillofac Surg       Date:  2014-08-11       Impact factor: 1.895

5.  Intravenous Pharmacokinetics, Local Tolerability, and Hemolysis of an SBE7-β-Cyclodextrin Formulation of the Neurokinin-1 Receptor Antagonist Vestipitant.

Authors:  Richard A Brigandi; Steven F Russ; Chantal Petit; Brendan Johnson; Scott Croy; Peter Hodsman; Fran Muller
Journal:  Clin Pharmacol Drug Dev       Date:  2014-05-26

Review 6.  Postoperative nausea and vomiting: A simple yet complex problem.

Authors:  Safiya Imtiaz Shaikh; D Nagarekha; Ganapati Hegade; M Marutheesh
Journal:  Anesth Essays Res       Date:  2016 Sep-Dec
  6 in total

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