Literature DB >> 20843983

Low allergenic potential with fondaparinux: results of a prospective investigation.

Marc Schindewolf1, Julia Scheuermann, Hartmut Kroll, Jurate Garbaraviciene, Carola Hecking, Ingo Marzi, Manfred Wolter, Roland Kaufmann, Wolf-Henning Boehncke, Edelgard Lindhoff-Last, Ralf J Ludwig.   

Abstract

OBJECTIVE: To determine the incidence and causes of skin reactions to the synthetic pentasaccharide fondaparinux. PATIENTS AND METHODS: Patients who received prophylactic/therapeutic subcutaneous fondaparinux treatment for more than 7 days were prospectively examined for cutaneous adverse effects between September 1, 2008, and April 30, 2009. When indicated, other procedures, such as skin biopsy, allergy testing, and clinical/laboratory assessment for thrombosis and heparin-induced thrombocytopenia, were performed.
RESULTS: Overall, 231 patients were enrolled. No patient developed typical delayed type IV hypersensitivity (DTH) erythematous skin lesions. However, one female patient experienced abdominal pruritus at sites of injection. Histology revealed a mild lymphohistiocytic infiltrate, confirming a DTH reaction. Heparin-induced thrombocytopenia, as another possible underlying pathomechanism for cutaneous lesions, was ruled out clinically and serologically. Hence, the overall incidence of fondaparinux-induced allergic skin lesions was 0.4% (95% confidence interval, 0.01%-2.4%). No cross-allergies were observed in patients with DTH reaction to heparins.
CONCLUSION: Fondaparinux has a low allergenic potential. The incidence of allergic cutaneous DTH reactions is almost 20 times lower compared to that with commonly used heparins. These results, together with the known low prevalence of secondary thrombotic events or heparin-induced thrombocytopenia during fondaparinux therapy, suggest that in selected patients fondaparinux might substantially improve patient care, therapeutic safety, and cost-effectiveness of anticoagulant therapy. TRIAL REGISTRATION: clinicaltrials.gov identifier: NCT00510432.

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Year:  2010        PMID: 20843983      PMCID: PMC2947963          DOI: 10.4065/mcp.2010.0346

Source DB:  PubMed          Journal:  Mayo Clin Proc        ISSN: 0025-6196            Impact factor:   7.616


  34 in total

1.  High rate of skin complications due to low-molecular-weight heparins in pregnant women.

Authors:  I Bank; E J Libourel; S Middeldorp; J Van Der Meer; H R Büller
Journal:  J Thromb Haemost       Date:  2003-04       Impact factor: 5.824

2.  Minor transplacental passage of fondaparinux in vivo.

Authors:  Carl-Erik H Dempfle
Journal:  N Engl J Med       Date:  2004-04-29       Impact factor: 91.245

3.  Intolerance of fondaparinux in a patient allergic to heparins.

Authors:  Katrin Hirsch; Ralf J Ludwig; Edelgard Lindhoff-Last; Roland Kaufmann; Wolf-Henning Boehncke
Journal:  Contact Dermatitis       Date:  2004-06       Impact factor: 6.600

4.  Tolerance to the synthetic pentasaccharide fondaparinux in heparin sensitization.

Authors:  C Sacher; N Hunzelmann
Journal:  Allergy       Date:  2003-12       Impact factor: 13.146

Review 5.  Chemical synthesis of glycosaminoglycans: new approaches to antithrombotic drugs.

Authors:  M Petitou; J C Lormeau; J Choay
Journal:  Nature       Date:  1991-04-18       Impact factor: 49.962

Review 6.  Heparin and low-molecular-weight heparin: mechanisms of action, pharmacokinetics, dosing, monitoring, efficacy, and safety.

Authors:  J Hirsh; T E Warkentin; S G Shaughnessy; S S Anand; J L Halperin; R Raschke; C Granger; E M Ohman; J E Dalen
Journal:  Chest       Date:  2001-01       Impact factor: 9.410

Review 7.  A synthetic antithrombin III binding pentasaccharide is now a drug! What comes next?

Authors:  Maurice Petitou; Constant A A van Boeckel
Journal:  Angew Chem Int Ed Engl       Date:  2004-06-14       Impact factor: 15.336

8.  Incidence and causes of heparin-induced skin lesions.

Authors:  Marc Schindewolf; Svantje Schwaner; Manfred Wolter; Hartmut Kroll; Andreas Recke; Roland Kaufmann; Wolf-Henning Boehncke; Edelgard Lindhoff-Last; Ralf J Ludwig
Journal:  CMAJ       Date:  2009-09-28       Impact factor: 8.262

9.  Fondaparinux: a suitable alternative in cases of delayed-type allergy to heparins and semisynthetic heparinoids? A study of 7 cases.

Authors:  U Jappe; U Juschka; N Kuner; B M Hausen; K Krohn
Journal:  Contact Dermatitis       Date:  2004-08       Impact factor: 6.600

10.  Antibodies from patients with heparin-induced thrombocytopenia/thrombosis are specific for platelet factor 4 complexed with heparin or bound to endothelial cells.

Authors:  G P Visentin; S E Ford; J P Scott; R H Aster
Journal:  J Clin Invest       Date:  1994-01       Impact factor: 14.808

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  2 in total

1.  Fondaparinux Pre-, Peri-, and/or Postpartum for the Prophylaxis/Treatment of Venous Thromboembolism (FondaPPP).

Authors:  Carl-Erik Dempfle; Jürgen Koscielny; Edelgard Lindhoff-Last; Birgit Linnemann; Irene Bux-Gewehr; Günther Kappert; Ute Scholz; Stefan Kropff; Sonja Eberle; Peter Bramlage; Andreas Heinken
Journal:  Clin Appl Thromb Hemost       Date:  2021 Jan-Dec       Impact factor: 2.389

2.  Sustained drug-related reaction with eosinophilia and systemic symptoms (DRESS) triggered by low molecular weight heparins in COVID-19: management and precision diagnosis.

Authors:  Elena Minenna; Nada Chaoul; Maria Pia Rossi; Lucia Giliberti; Marcello Albanesi; Eustachio Nettis; Maria Pia Foschino Barbaro; Danilo Di Bona; Maria Filomena Caiaffa; Luigi Macchia
Journal:  Postepy Dermatol Alergol       Date:  2021-10-01       Impact factor: 1.664

  2 in total

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