Literature DB >> 20807345

A novel 12-week study, with three randomized, double-blind placebo-controlled periods to evaluate fentanyl buccal tablets for the relief of breakthrough pain in opioid-tolerant patients with noncancer-related chronic pain.

John T Farrar1, John Messina, Fang Xie, Russell K Portenoy.   

Abstract

OBJECTIVE: To evaluate the time of onset, overall efficacy, and safety of fentanyl buccal tablet (FBT) for noncancer-related breakthrough pain (BTP) in opioid-tolerant adults over 12 weeks.
DESIGN: A novel 12-week study that mimicked clinical practice with dose titration to effective dose, open-label treatment, and three randomized, double-blind, placebo-controlled, multiple-crossover periods at weeks 4, 8, and 12. For each double-blind period, study patients received nine doses (FBT = 6, placebo = 3) in a randomized sequence.
SETTING: Twenty-one study centers in the United States. POPULATION: Opioid-tolerant adults with noncancer-related chronic pain and BTP. OUTCOME MEASURES: The primary outcome was the sum of the pain intensity differences (PID) 5-60 minutes post dose (SPID₆₀) during the final double-blind period. Secondary outcomes included pain relief (PR), meaningful PR, and proportion of episodes with a PID of ≥33% and ≥50%.
RESULTS: Of 148 patients who entered the titration phase, 105 (71%) achieved a successful dose and 81 (55%) participated in all three assessment periods in the study. The final RCT assessment period results demonstrated continued efficacy of FBT vs placebo (P < 0.05) for SPID₆₀ (mean [SD]: 7.7 [6.2] vs 4.6 [4.7]). The average onset of PR began at 5 minutes, with meaningful PR by ≤10 minutes. The proportion of episodes with ≥33% improvement in PI was 7% with FBT vs 3% with placebo at 5 minutes and with ≥50% was 17% vs 10% at 15 minutes. All periods showed similar results. Adverse events and patient discontinuations were generally typical of clinical opioid use.
CONCLUSIONS: FBT showed continued clinically important analgesic effects and was generally well tolerated over 12 weeks of treatment. Wiley Periodicals, Inc.

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Year:  2010        PMID: 20807345     DOI: 10.1111/j.1526-4637.2010.00939.x

Source DB:  PubMed          Journal:  Pain Med        ISSN: 1526-2375            Impact factor:   3.750


  8 in total

Review 1.  [Chronic non-cancer-related pain. Long-term treatment with rapid-release and short-acting opioids in the context of misuse and dependency].

Authors:  R Scharnagel; U Kaiser; A Schütze; R Heineck; G Gossrau; R Sabatowski
Journal:  Schmerz       Date:  2013-02       Impact factor: 1.107

2.  Efficacy and safety of sublingual fentanyl orally disintegrating tablets in patients with breakthrough pain: multicentre prospective study.

Authors:  Jordi Guitart; Isabel Vargas; Vicente De Sanctis; Julia Ferreras; Jose Fuentes; Rafael Salazar; Juan M Vázquez; Jordi Folch; Jordi Moya; Hermann Ribera; Francisco Rodelas; Albert Tomás; María Arilla; Joan Coma; Teresa Aberasturi; Dolores Sintes; Ester Lombán
Journal:  Clin Drug Investig       Date:  2013-09       Impact factor: 2.859

3.  Differential development of antinociceptive tolerance to morphine and fentanyl is not linked to efficacy in the ventrolateral periaqueductal gray of the rat.

Authors:  Erin N Bobeck; Rachel A Haseman; Dana Hong; Susan L Ingram; Michael M Morgan
Journal:  J Pain       Date:  2012-07-03       Impact factor: 5.820

Review 4.  Analysis of opioid efficacy, tolerance, addiction and dependence from cell culture to human.

Authors:  Michael M Morgan; MacDonald J Christie
Journal:  Br J Pharmacol       Date:  2011-10       Impact factor: 8.739

5.  [Use of rapid-onset fentanyl preparations beyond indication : A random questionnaire survey among congress participants and pain physicians].

Authors:  Stefan Wirz; Michael Schenk; Hannes Hofbauer; Hans-Christian Wartenberg; Marco Cascella; Kristin Kieselbach
Journal:  Schmerz       Date:  2020-09-25       Impact factor: 1.107

6.  Chronic inflammatory pain prevents tolerance to the antinociceptive effect of morphine microinjected into the ventrolateral periaqueductal gray of the rat.

Authors:  Melissa L Mehalick; Susan L Ingram; Sue A Aicher; Michael M Morgan
Journal:  J Pain       Date:  2013-10-22       Impact factor: 5.820

Review 7.  A comprehensive review of rapid-onset opioids for breakthrough pain.

Authors:  Howard Smith
Journal:  CNS Drugs       Date:  2012-06-01       Impact factor: 5.749

8.  Considerations in selecting rapid-onset opioids for the management of breakthrough pain.

Authors:  Howard S Smith
Journal:  J Pain Res       Date:  2013-03-06       Impact factor: 3.133

  8 in total

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