Literature DB >> 20717823

Functional oestrogen receptor α imaging in endometrial carcinoma using 16α-[¹⁸F]fluoro-17β-oestradiol PET.

Tetsuya Tsujikawa1, Yoshio Yoshida, Yasushi Kiyono, Tetsuji Kurokawa, Takashi Kudo, Yasuhisa Fujibayashi, Fumikazu Kotsuji, Hidehiko Okazawa.   

Abstract

PURPOSE: To investigate the correlation between uptake of 16α-[(18)F]fluoro-17β-oestradiol (FES) and expression of oestrogen receptors as well as other related immunohistochemistry markers, positron emission tomography (PET) was performed in patients with endometrial carcinoma before surgery.
METHODS: Nineteen patients with endometrioid adenocarcinoma underwent preoperative PET studies with FES and 2-[(18)F]fluoro-2-deoxy-D: -glucose (FDG). Standardized uptake values (SUVs) for each tracer and the regional FDG to FES SUV ratio were calculated using images after coregistration. PET values were compared with postoperative stage, differentiation grade and immunohistochemical scores including oestrogen receptor subtypes (ERα, ERβ), progesterone receptor B (PR-B), Ki-67 and glucose transporter 1 (GLUT1).
RESULTS: FES uptake showed a significantly positive correlation with expression of ERα. The FDG to FES ratio showed a significantly negative correlation with expression of ERα and PR-B. The FES uptake and FDG to FES ratio did not correlate with expression of ERβ, Ki-67 or GLUT1. FDG uptake was not correlated with any of the immunohistochemical scores. The PR-B score was strongly correlated with the ERα score. Well-differentiated carcinoma (grade 1) showed a significantly higher FES uptake and significantly lower FDG to FES ratio than moderately or poorly differentiated carcinoma (grade 2-3). None of the PET parameters were significantly different between advanced-stage carcinoma (≥ stage IB) and early-stage carcinoma (IA) based on the Féderation International de Gynécologie et d'Obstétrique (FIGO) staging classification. Differentiation grade was the most closely correlated parameter to FES uptake and FDG to FES ratio by multivariate analyses.
CONCLUSION: FES PET combined with FDG would be useful for non-invasive evaluation of ERα distribution, as well as ERα function, which reflects differentiation grade in endometrial carcinoma.

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Year:  2010        PMID: 20717823     DOI: 10.1007/s00259-010-1589-8

Source DB:  PubMed          Journal:  Eur J Nucl Med Mol Imaging        ISSN: 1619-7070            Impact factor:   9.236


  37 in total

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Review 2.  Transcription activation by estrogen and progesterone receptors.

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5.  Quantitative imaging of estrogen receptor expression in breast cancer with PET and 18F-fluoroestradiol.

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7.  Uterine tumors: pathophysiologic imaging with 16alpha-[18F]fluoro-17beta-estradiol and 18F fluorodeoxyglucose PET--initial experience.

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8.  Automatic synthesis of 16 alpha-[(18)F]fluoro-17beta-estradiol using a cassette-type [(18)F]fluorodeoxyglucose synthesizer.

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10.  Oestrogen receptor beta expression and depth of myometrial invasion in human endometrial cancer.

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  14 in total

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2.  Additional value of 16α-[18F]fluoro-17β-oestradiol PET for differential diagnosis between uterine sarcoma and leiomyoma in patients with positive or equivocal findings on [18F]fluorodeoxyglucose PET.

Authors:  Yoshio Yoshida; Yasushi Kiyono; Tetsuya Tsujikawa; Tetsuji Kurokawa; Hidehiko Okazawa; Fumikazu Kotsuji
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3.  Linked Hexokinase and Glucose-6-Phosphatase Activities Reflect Grade of Ovarian Malignancy.

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4.  Oestrogen-related tumour phenotype: positron emission tomography characterisation with ¹⁸F-FDG and ¹⁸F-FES.

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5.  Improved Estrogen Receptor Assessment by PET Using the Novel Radiotracer 18F-4FMFES in Estrogen Receptor-Positive Breast Cancer Patients: An Ongoing Phase II Clinical Trial.

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6.  Assessment of the novel estrogen receptor PET tracer 4-fluoro-11β-methoxy-16α-[(18)F]fluoroestradiol (4FMFES) by PET imaging in a breast cancer murine model.

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Review 8.  What's New in Imaging for Gynecologic Cancer?

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9.  PET Imaging of Estrogen Receptors Using 18F-Based Radioligands.

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10.  Prognostic Value of 16α-18F-Fluoro-17β-Estradiol PET as a Predictor of Disease Outcome in Endometrial Cancer: A Prospective Study.

Authors:  Shizuka Yamada; Hideaki Tsuyoshi; Makoto Yamamoto; Tetsuya Tsujikawa; Yasushi Kiyono; Hidehiko Okazawa; Yoshio Yoshida
Journal:  J Nucl Med       Date:  2020-10-02       Impact factor: 10.057

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