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15 in total

1. THE CHANGES IN RESPONSE AND IN IONIC CONTENT OF SMOOTH MUSCLE PRODUCED BY ACETYLCHOLINE ACTON AND BY CALCIUM DEFICIENCY.

Authors: W D PATON; A M ROTHSCHILD
Journal: Br J Pharmacol Chemother Date: 1965-04

2. Dissociation constants and relative efficacies of agonists acting on alpha adrenergic receptors in rabbit aorta.

Authors: J C Besse; R F Furchgott
Journal: J Pharmacol Exp Ther Date: 1976-04 Impact factor: 4.030

3. Analysis of dose-response curves and calculation of agonist dissociation constants using a weighted nonlinear curve fitting program.

Authors: G A McPherson; P Molenaar; C Raper; E Malta
Journal: J Pharmacol Methods Date: 1983-12

4. Operational models of pharmacological agonism.

Authors: J W Black; P Leff
Journal: Proc R Soc Lond B Biol Sci Date: 1983-12-22

5. Pharmacological estimation of drug-receptor dissociation constants. Statistical evaluation. I. Agonists.

Authors: R B Parker; D R Waud
Journal: J Pharmacol Exp Ther Date: 1971-04 Impact factor: 4.030

6. The affinity and efficacy of onium salts on the frog rectus abdominis.

Authors: R B Barlow; N C Scott; R P Stephenson
Journal: Br J Pharmacol Chemother Date: 1967-09

7. Use of selective antagonists for determining the types of receptors mediating the actions of 5-hydroxytryptamine and tryptamine in the isolated rabbit aorta.

Authors: J S Stollak; R F Furchgott
Journal: J Pharmacol Exp Ther Date: 1983-01 Impact factor: 4.030

8. Noradrenergic component in the vasoconstriction induced by 5-hydroxytryptamine in goat cerebral arteries.

Authors: J Marin; M Salaices; B Gómez; S Lluch
Journal: J Pharm Pharmacol Date: 1981-11 Impact factor: 3.765

9. Mechanism of the indirect sympathomimetic effect of 5-hydroxytrypt-amine on the isolated heart of the rabbit.

Authors: J R Fozard; G M Mwaluko
Journal: Br J Pharmacol Date: 1976-05 Impact factor: 8.739

10. Receptors for 5-hydroxytryptamine and noradrenaline in rabbit isolated ear artery and aorta.

Authors: E Apperley; P P Humphrey; G P Levy
Journal: Br J Pharmacol Date: 1976-10 Impact factor: 8.739

5 in total

1. 15-Keto-PGE₂ acts as a biased/partial agonist to terminate PGE₂-evoked signaling.

Authors: Suzu Endo; Akiko Suganami; Keijo Fukushima; Kanaho Senoo; Yumi Araki; John W Regan; Masato Mashimo; Yutaka Tamura; Hiromichi Fujino
Journal: J Biol Chem Date: 2020-07-29 Impact factor: 5.157

Review 2. Finding the Perfect Fit: Conformational Biosensors to Determine the Efficacy of GPCR Ligands.

Authors: Keith M Olson; Andra Campbell; Andrew Alt; John R Traynor
Journal: ACS Pharmacol Transl Sci Date: 2022-08-14

3. A single amino acid substitution in CXCL12 confers functional selectivity at the beta-arrestin level.

Authors: Antonella Rigo; Isacco Ferrarini; Giulio Innamorati; Fabrizio Vinante
Journal: Oncotarget Date: 2018-06-22

4. The Gαs-protein-mediated pathway may be steadily stimulated by prostanoid EP2 receptors, but not by EP4 receptors.

Authors: Keijo Fukushima; Kanaho Senoo; Naoki Kurata; John W Regan; Hiromichi Fujino
Journal: FEBS Open Bio Date: 2022-02-15 Impact factor: 2.693

5. In vivo and in vitro Characterization of a Partial Mu Opioid Receptor Agonist, NKTR-181, Supports Future Therapeutic Development.

Authors: Alex S Lee; Suchi Tiwari; Isabel Bishop; Vartan Matossian; Nicole Romaneschi; Takahiro Miyazaki; Laurie VanderVeen; Jonathan Zalevsky; Kathryn DeFea; Catherine M Cahill; Wendy M Walwyn
Journal: Front Pain Res (Lausanne) Date: 2021-08-23

5 in total