Literature DB >> 20584608

Antimalarial 3-arylamino-6-benzylamino-1,2,4,5-tetrazines.

Duong Nhu1, Sandra Duffy, Vicky M Avery, Andrew Hughes, Jonathan B Baell.   

Abstract

We report on novel 3-arylamino-6-benzylamino-1,2,4,5-tetrazines with potent activity against Plasmodium falciparum. Copyright 2010 Elsevier Ltd. All rights reserved.

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Year:  2010        PMID: 20584608     DOI: 10.1016/j.bmcl.2010.06.036

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN: 0960-894X            Impact factor:   2.823


  4 in total

1.  Phenyl Ether- and Aniline-Containing 2-Aminoquinolines as Potent and Selective Inhibitors of Neuronal Nitric Oxide Synthase.

Authors:  Maris A Cinelli; Huiying Li; Anthony V Pensa; Soosung Kang; Linda J Roman; Pavel Martásek; Thomas L Poulos; Richard B Silverman
Journal:  J Med Chem       Date:  2015-10-27       Impact factor: 7.446

2.  Trifunctional cross-linker for mapping protein-protein interaction networks and comparing protein conformational states.

Authors:  Dan Tan; Qiang Li; Mei-Jun Zhang; Chao Liu; Chengying Ma; Pan Zhang; Yue-He Ding; Sheng-Bo Fan; Li Tao; Bing Yang; Xiangke Li; Shoucai Ma; Junjie Liu; Boya Feng; Xiaohui Liu; Hong-Wei Wang; Si-Min He; Ning Gao; Keqiong Ye; Meng-Qiu Dong; Xiaoguang Lei
Journal:  Elife       Date:  2016-03-08       Impact factor: 8.140

3.  DFT-based reactivity and combined QSAR, molecular docking of 1,2,4,5-Tetrazine derivatives as inhibitors of Pim-1 kinase.

Authors:  Halima Hazhazi; Nadjib Melkemi; Toufik Salah; Mohammed Bouachrine
Journal:  Heliyon       Date:  2019-09-26

4.  ZGDHu-1 for cancer therapy.

Authors:  Jinlin Liu; Liannv Qiu; Jun Xia; Sufeng Chen; Xiping Yu; Yonglie Zhou
Journal:  Oncol Lett       Date:  2017-09-28       Impact factor: 2.967

  4 in total

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