Literature DB >> 20564576

Hit identification and biological evaluation of anticancer pyrazolopyrimidines endowed with anti-inflammatory activity.

Stefano Alcaro1, Anna Artese, Maurizio Botta, Alessandra T Zizzari, Francisco Orallo, Francesco Ortuso, Silvia Schenone, Chiara Brullo, Matilde Yáñez.   

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Year:  2010        PMID： 20564576     DOI： 10.1002/cmdc.201000165

Source DB:  PubMed          Journal:  ChemMedChem        ISSN： 1860-7179            Impact factor:   3.466


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  5 in total

1.  A facile, regioselective synthesis of novel 3-(N-phenylcarboxamide)pyrazolo[1,5-a]pyrimidine analogs in the presence of KHSO4 in aqueous media assisted by ultrasound and their antibacterial activities.

Authors:  Shunan Kaping; Ivee Boiss; Laishram Indira Singha; Philippe Helissey; Jai N Vishwakarma
Journal:  Mol Divers       Date:  2015-10-28       Impact factor: 2.943

2.  A facile environment-friendly one-pot two-step regioselective synthetic strategy for 3,7-diarylpyrazolo[1,5-a]pyrimidines related to zaleplon and 3,6-diarylpyrazolo[1,5-a]pyrimidine-7-amines assisted by KHSO₄ in aqueous media.

Authors:  Asem Satyapati Devi; Shunan Kaping; Jai Narain Vishwakarma
Journal:  Mol Divers       Date:  2015-05-28       Impact factor: 2.943

3.  Synthesis, Structural Elucidation, and In Vitro Antitumor Activities of Some Pyrazolopyrimidines and Schiff Bases Derived from 5-Amino-3-(arylamino)-1H-pyrazole-4-carboxamides.

Authors:  Taghrid S Hafez; Souad A Osman; Hisham Abdallah A Yosef; Amira S Abd El-All; Ashraf S Hassan; Abdallah A El-Sawy; Mohamed M Abdallah; Mahmoud Youns
Journal:  Sci Pharm       Date:  2013-01-03

4.  18F-labeled pyrazolo[1,5-a]pyrimidine derivatives: synthesis from 2,4-dinitrobenzamide and tosylate precursors and comparative biological evaluation for tumor imaging with positron emission tomography.

Authors:  Jingli Xu; Hang Liu; Guixia Li; Yong He; Rui Ding; Xiao Wang; Man Feng; Shuting Zhang; Yurong Chen; Shilei Li; Mingxia Zhao; Yingruo Li; Chuanmin Qi; Yonghong Dang
Journal:  Molecules       Date:  2012-03-27       Impact factor: 4.411

5.  Synthesis, Characterization, and Cytotoxicity of Some New 5-Aminopyrazole and Pyrazolo[1,5-a]pyrimidine Derivatives.

Authors:  Ashraf S Hassan; Taghrid S Hafez; Souad A Osman
Journal:  Sci Pharm       Date:  2014-10-24
  5 in total

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