Literature DB >> 20514155

Canadian consensus guidelines for the optimal use of etravirine in the treatment of HIV-infected adults.

Marianne Harris1, Jonathan B Angel, Jean-Guy Baril, Anita Rachlis, Benoit Trottier.   

Abstract

BACKGROUND AND OBJECTIVES: A group of five Canadian physicians with significant experience in HIV management was convened. Their goal was to develop guidance specifically for Canadian HIV-treating physicians on the appropriate use of etravirine (TMC125, Intelence, Tibotec BVBA, Belgium) in adult HIV-infected patients.
METHODS: Evidence from the published literature, conference presentations and expert opinions of the group members were used to develop the recommendations. Feedback on the draft recommendations was obtained from this core group, and from seven other physicians across Canada with clinical HIV treatment expertise and experience in the use of etravirine, as well as two Canadian scientists with HIV expertise. The final recommendations represent the core group's consensus agreement, taking all feedback into consideration. RESULTS AND
CONCLUSIONS: The recommendations were developed to guide physicians in the optimal use of etravirine. The issues considered included HIV disease status, antiretroviral treatment history, drug resistance profiles, predictors of response to etravirine, background antiretroviral regimen and drug-drug interactions.

Entities:  

Keywords:  Etravirine; HIV; NNRTI; Recommendations; Resistance; TMC125; Treatment

Year:  2009        PMID: 20514155      PMCID: PMC2706403          DOI: 10.1155/2009/658125

Source DB:  PubMed          Journal:  Can J Infect Dis Med Microbiol        ISSN: 1712-9532            Impact factor:   2.471


  31 in total

1.  Pharmacokinetic and pharmacodynamic study of the concomitant administration of methadone and TMC125 in HIV-negative volunteers.

Authors:  Monika Schöller-Gyüre; Wim van den Brink; Thomas N Kakuda; Brian Woodfall; Goedele De Smedt; Hilde Vanaken; Tanja Stevens; Monika Peeters; Kati Vandermeulen; Richard M W Hoetelmans
Journal:  J Clin Pharmacol       Date:  2008-01-14       Impact factor: 3.126

Review 2.  Update of the drug resistance mutations in HIV-1: 2007.

Authors:  Victoria A Johnson; Françoise Brun-Vézinet; Bonaventura Clotet; Huldrych F Günthard; Daniel R Kuritzkes; Deenan Pillay; Jonathan M Schapiro; Douglas D Richman
Journal:  Top HIV Med       Date:  2007 Aug-Sep

3.  Durable efficacy of tipranavir-ritonavir in combination with an optimised background regimen of antiretroviral drugs for treatment-experienced HIV-1-infected patients at 48 weeks in the Randomized Evaluation of Strategic Intervention in multi-drug reSistant patients with Tipranavir (RESIST) studies: an analysis of combined data from two randomised open-label trials.

Authors:  Charles B Hicks; Pedro Cahn; David A Cooper; Sharon L Walmsley; Christine Katlama; Bonaventura Clotet; Adriano Lazzarin; Margaret A Johnson; Dietmar Neubacher; Douglas Mayers; Hernan Valdez
Journal:  Lancet       Date:  2006-08-05       Impact factor: 79.321

4.  TMC125, a novel next-generation nonnucleoside reverse transcriptase inhibitor active against nonnucleoside reverse transcriptase inhibitor-resistant human immunodeficiency virus type 1.

Authors:  Koen Andries; Hilde Azijn; Theo Thielemans; Donald Ludovici; Michael Kukla; Jan Heeres; Paul Janssen; Bart De Corte; Johan Vingerhoets; Rudi Pauwels; Marie-Pierre de Béthune
Journal:  Antimicrob Agents Chemother       Date:  2004-12       Impact factor: 5.191

5.  Evaluating the role of etravirine in the second-line antiretroviral therapy after failing an initial non-nucleoside reverse transcriptase inhibitor-based regimen in a resource-limited setting.

Authors:  Somnuek Sungkanuparph; Weerawat Manosuthi; Sasisopin Kiertiburanakul; Bucha Piyavong; Wasun Chantratita
Journal:  Curr HIV Res       Date:  2008-09       Impact factor: 1.581

6.  Roles of conformational and positional adaptability in structure-based design of TMC125-R165335 (etravirine) and related non-nucleoside reverse transcriptase inhibitors that are highly potent and effective against wild-type and drug-resistant HIV-1 variants.

Authors:  Kalyan Das; Arthur D Clark; Paul J Lewi; Jan Heeres; Marc R De Jonge; Lucien M H Koymans; H Maarten Vinkers; Frederik Daeyaert; Donald W Ludovici; Michael J Kukla; Bart De Corte; Robert W Kavash; Chih Y Ho; Hong Ye; Mark A Lichtenstein; Koen Andries; Rudi Pauwels; Marie-Pierre De Béthune; Paul L Boyer; Patrick Clark; Stephen H Hughes; Paul A J Janssen; Eddy Arnold
Journal:  J Med Chem       Date:  2004-05-06       Impact factor: 7.446

7.  Successful rescue therapy with Raltegravir (MK-0518) and Etravirine (TMC125) in an hiv-infected patient failing all four classes of antiretroviral drugs.

Authors:  Antonio Di Biagio; Bianca Bruzzone; Raffaella Rosso; Ottavia Viganò; Giancarlo Icardi; Claudio Viscoli; Stefano Rusconi
Journal:  AIDS Patient Care STDS       Date:  2008-05       Impact factor: 5.078

8.  Efficacy and safety of etravirine (TMC125) in patients with highly resistant HIV-1: primary 24-week analysis.

Authors:  Jeffrey P Nadler; Daniel S Berger; Gary Blick; Paul J Cimoch; Calvin J Cohen; Richard N Greenberg; Charles B Hicks; Richard M W Hoetelmans; Kathy J Iveson; Dushyantha S Jayaweera; Anthony M Mills; Monika P Peeters; Peter J Ruane; Peter Shalit; Shannon R Schrader; Stephen M Smith; Corklin R Steinhart; Melanie Thompson; Johan H Vingerhoets; Ellen Voorspoels; Douglas Ward; Brian Woodfall
Journal:  AIDS       Date:  2007-03-30       Impact factor: 4.177

Review 9.  TMC-125 Tibotec.

Authors:  Bernhard A Haslinger; Gabriele Arendt
Journal:  Curr Opin Investig Drugs       Date:  2004-02

10.  Potent nonnucleoside reverse transcriptase inhibitors target HIV-1 Gag-Pol.

Authors:  Anna Figueiredo; Katie L Moore; Johnson Mak; Nicolas Sluis-Cremer; Marie-Pierre de Bethune; Gilda Tachedjian
Journal:  PLoS Pathog       Date:  2006-11       Impact factor: 6.823

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