Literature DB >> 20486935

Synthesis and antifungal activities of new pyrazole derivatives via 1,3-dipolar cycloaddition reaction.

Chuan-Yu Zhang1, Xing-Hai Liu, Bao-Lei Wang, Su-Hua Wang, Zheng-Ming Li.   

Abstract

A series of cycloadducts--pyrazoles via 1,3-dipolar cycloaddition reactions of generated nitrilimines with N-(4-chloro-2-fluorophenyl)maleimide were described. The novel compounds synthesized were characterized by (1)H NMR, MS, and elemental analysis. The fungicidal tests showed that most of the title compounds exhibit significant fungicidal activities against Corynespora cassiicola.

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Year:  2010        PMID： 20486935     DOI： 10.1111/j.1747-0285.2010.00948.x

Source DB:  PubMed          Journal:  Chem Biol Drug Des        ISSN： 1747-0277            Impact factor:   2.817


  5 in total

1.  Crystal structure of (4Z)-4-[(di-methyl-amino)-methyl-idene]-3,5-dioxo-2-phenyl-pyrazolidine-1-carbaldehyde.

Authors:  Joel T Mague; Shaaban K Mohamed; Mehmet Akkurt; Eman A Ahmed; Ahmed Khodairy
Journal:  Acta Crystallogr E Crystallogr Commun       Date:  2015-06-03

2.  Novel Antimicrobial Agents: Fluorinated 2-(3-(Benzofuran-2-yl) pyrazol-1-yl)thiazoles.

Authors:  Hanan A Mohamed; Ehab Abdel-Latif; Bakr F Abdel-Wahab; Ghada E A Awad
Journal:  Int J Med Chem       Date:  2013-09-11

3.  Discovery of Potent VEGFR-2 Inhibitors based on Furopyrimidine and Thienopyrimidne Scaffolds as Cancer Targeting Agents.

Authors:  Marwa A Aziz; Rabah A T Serya; Deena S Lasheen; Amal Kamal Abdel-Aziz; Ahmed Esmat; Ahmed M Mansour; Abdel Nasser B Singab; Khaled A M Abouzid
Journal:  Sci Rep       Date:  2016-04-15       Impact factor: 4.379

4.  Sc(OTf)3-Mediated [4 + 2] Annulations of N-Carbonyl Aryldiazenes with Cyclopentadiene to Construct Cinnoline Derivatives: Azo-Povarov Reaction.

Authors:  Xabier Jiménez-Aberásturi; Francisco Palacios; Jesús M de Los Santos
Journal:  J Org Chem       Date:  2022-08-16       Impact factor: 4.198

5.  Synergistic antifungal effect of cyclized chalcone derivatives and fluconazole against Candida albicans.

Authors:  Aijaz Ahmad; Mohmmad Younus Wani; Mrudula Patel; Abilio J F N Sobral; Adriano G Duse; Faisal Mohammed Aqlan; Abdullah Saad Al-Bogami
Journal:  Medchemcomm       Date:  2017-10-17       Impact factor: 3.597
  5 in total

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