Literature DB >> 20445575

Synergistic activity of the Src/Abl inhibitor bosutinib in combination with imatinib.

S Redaelli, F Boschelli, P Perini, A Pirola, M Viltadi, C Gambacorti-Passerini.   

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Year:  2010        PMID: 20445575     DOI: 10.1038/leu.2010.79

Source DB:  PubMed          Journal:  Leukemia        ISSN: 0887-6924            Impact factor:   11.528


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  10 in total

1.  Long-term treatment with bosutinib in a phase 1/2 study in Japanese chronic myeloid leukemia patients resistant/intolerant to prior tyrosine kinase inhibitor treatment.

Authors:  Naoto Takahashi; Chiaki Nakaseko; Yukio Kobayashi; Koichi Miyamura; Chiho Ono; Yuichiro Koide; Yosuke Fujii; Kazunori Ohnishi
Journal:  Int J Hematol       Date:  2017-04-13       Impact factor: 2.490

2.  Aberrant signalling by protein kinase CK2 in imatinib-resistant chronic myeloid leukaemia cells: biochemical evidence and therapeutic perspectives.

Authors:  Christian Borgo; Luca Cesaro; Valentina Salizzato; Maria Ruzzene; Maria Lina Massimino; Lorenzo A Pinna; Arianna Donella-Deana
Journal:  Mol Oncol       Date:  2013-08-22       Impact factor: 6.603

3.  Chronic myeloid leukemia 2011: successes, challenges, and strategies--proceedings of the 5th annual BCR-ABL1 positive and BCR-ABL1 negative myeloproliferative neoplasms workshop.

Authors:  Tariq I Mughal; Jerald P Radich; Richard A Van Etten; Alfonso Quintás-Cardama; Tomasz Skorski; Farhad Ravandi; Daniel J DeAngelo; Carlo Gambacorti-Passerini; Giovanni Martinelli; Ayalew Tefferi
Journal:  Am J Hematol       Date:  2011-09       Impact factor: 10.047

4.  A kinase profile-adapted drug combination elicits synergistic cooperative effects on leukemic cells carrying BCR-ABL1T315I in Ph+ CML.

Authors:  Karoline V Gleixner; Irina Sadovnik; Mathias Schneeweiss; Gregor Eisenwort; Konstantin Byrgazov; Gabriele Stefanzl; Daniela Berger; Harald Herrmann; Emir Hadzijusufovic; Thomas Lion; Peter Valent
Journal:  Leuk Res       Date:  2018-12-28       Impact factor: 3.156

5.  Effects of the CK2 inhibitors CX-4945 and CX-5011 on drug-resistant cells.

Authors:  Sofia Zanin; Christian Borgo; Cristina Girardi; Sean E O'Brien; Yoshihiko Miyata; Lorenzo A Pinna; Arianna Donella-Deana; Maria Ruzzene
Journal:  PLoS One       Date:  2012-11-08       Impact factor: 3.240

Review 6.  Hematopoietic cell kinase (HCK) as a therapeutic target in immune and cancer cells.

Authors:  Ashleigh R Poh; Robert J J O'Donoghue; Matthias Ernst
Journal:  Oncotarget       Date:  2015-06-30

7.  Inhibition of protein kinase CK2 by CX-5011 counteracts imatinib-resistance preventing rpS6 phosphorylation in chronic myeloid leukaemia cells: new combined therapeutic strategies.

Authors:  Valentina Salizzato; Christian Borgo; Luca Cesaro; Lorenzo A Pinna; Arianna Donella-Deana
Journal:  Oncotarget       Date:  2016-04-05

8.  Factors influencing long-term efficacy and tolerability of bosutinib in chronic phase chronic myeloid leukaemia resistant or intolerant to imatinib.

Authors:  Tim H Brümmendorf; Jorge E Cortes; Hanna J Khoury; Hagop M Kantarjian; Dong-Wook Kim; Philippe Schafhausen; Maureen G Conlan; Mark Shapiro; Kathleen Turnbull; Eric Leip; Carlo Gambacorti-Passerini; Jeff H Lipton
Journal:  Br J Haematol       Date:  2015-11-04       Impact factor: 6.998

9.  Synergistic activity of ALK and mTOR inhibitors for the treatment of NPM-ALK positive lymphoma.

Authors:  Sara Redaelli; Monica Ceccon; Laura Antolini; Roberta Rigolio; Alessandra Pirola; Marco Peronaci; Carlo Gambacorti-Passerini; Luca Mologni
Journal:  Oncotarget       Date:  2016-11-08

10.  In Vitro Comparison of the Effects of Imatinib and Ponatinib on Chronic Myeloid Leukemia Progenitor/Stem Cell Features.

Authors:  Ignazia Tusa; Giulia Cheloni; Martina Poteti; Angela Silvano; Alessandro Tubita; Zoe Lombardi; Antonella Gozzini; Roberto Caporale; Barbara Scappini; Persio Dello Sbarba; Elisabetta Rovida
Journal:  Target Oncol       Date:  2020-10       Impact factor: 4.493

  10 in total

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