Literature DB >> 20404975

Sunitinib causes macrocytosis in patients with advanced renal cell carcinoma.

J Price1, R Shaarbaf, L Wood.   

Abstract

BACKGROUND: Sunitinib is approved for treatment of advanced renal cell carcinoma (RCC). Based on a clinical observation that patients receiving sunitinib developed macrocytosis, we undertook a study to further define this observation.
METHODS: In a retrospective review of RCC patients treated at a single centre, data on treatment duration, hematology parameters, concomitant medications, vitamin B₁₂and folate levels, and thyroid function were recorded.
RESULTS: The 43 patients reviewed had received a median of 5 cycles of sunitinib. Overall, 21 patients (49%) developed macrocytosis after a median of 3 cycles. Of the 9 patients that received 2 or fewer cycles, none developed macrocytosis. Among patients with macrocytosis, 9 (43%) had anemia at the time macrocytosis was first documented. In patients who did not develop macrocytosis, 82% showed a trend of increasing mean corpuscular volume.
CONCLUSIONS: Treatment with sunitinib in patients with RCC can cause macrocytosis. The frequency of macrocytosis increases with duration of treatment. The mechanism of sunitinib-associated macrocytosis remains to be elucidated.

Entities:  

Keywords:  Renal cell carcinoma; macrocytosis; sunitinib

Year:  2010        PMID: 20404975      PMCID: PMC2854633          DOI: 10.3747/co.v17i2.470

Source DB:  PubMed          Journal:  Curr Oncol        ISSN: 1198-0052            Impact factor:   3.677


  9 in total

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  4 in total

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