Literature DB >> 20377273

Total synthesis of (+/-)-galanthamine via a C3-selective Stille coupling and IMDA cycloaddition cascade of 3,5-dibromo-2-pyrone.

Jay Hyok Chang1, Ho-Ung Kang, In-Hak Jung, Cheon-Gyu Cho.   

Abstract

A new efficient synthetic route to (+/-)-galanthamine was devised by using a tandem C3-selective Stille coupling-IMDA cascade of 3,5-dibromo-2-pyrone as a key strategy.

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Year:  2010        PMID： 20377273     DOI： 10.1021/ol100617u

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  4 in total

1.  Regioselective Iodination of Chlorinated Aromatic Compounds Using Silver Salts.

Authors:  Sudhir N Joshi; Sandhya M Vyas; Huimin Wu; Michael W Duffel; Sean Parkin; Hans-Joachim Lehmler
Journal:  Tetrahedron       Date:  2011-09-30       Impact factor: 2.457

Review 2.  Recent advances in the synthesis of 2-pyrones.

Authors:  Jong Seok Lee
Journal:  Mar Drugs       Date:  2015-03-23       Impact factor: 5.118

Review 3.  Assessment on facile Diels-Alder approach of α-pyrone and terpenoquinone for the expedient synthesis of various natural scaffolds.

Authors:  Aluru Rammohan; Albert F Khasanov; Dmitry S Kopchuk; Duvvuru Gunasekar; Grigory V Zyryanov; Oleg N Chupakhin
Journal:  Nat Prod Bioprospect       Date:  2022-03-31

4.  Production of benzazepine derivatives via four-component reaction of isatins: study of antioxidant activity.

Authors:  Fathali Gholami Orimi; Behrooz Mirza; Zinatossadat Hossaini
Journal:  Mol Divers       Date:  2020-06-10       Impact factor: 2.943
  4 in total

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