Literature DB >> 20346668

Design, synthesis, and antibiofilm activity of 2-arylimino-3-aryl-thiazolidine-4-ones.

Bin Pan1, Ren-Zheng Huang, Shi-Qing Han, Di Qu, Ming-Li Zhu, Ping Wei, Han-Jie Ying.   

Abstract

A series of novel 2-arylimino-3-aryl-thiazolidine-4-ones was designed, synthesized and tested for in vitro antibiofilm activity against Staphylococcus epidermidis. Among them tested, some compounds with carboxylic acid groups showed good antibiofilm activity. The antibiofilm concentration of 1x was 6.25 microM. The structure-activity relationships revealed that incorporation of 2-phenylfuran moiety could greatly enhance antibiofilm activity of thiazolidine-4-one. Copyright 2010 Elsevier Ltd. All rights reserved.

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Year:  2010        PMID： 20346668     DOI： 10.1016/j.bmcl.2010.03.013

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  6 in total

Review 1.  Synthesis of histidine kinase inhibitors and their biological properties.

Authors:  Miyanou Rosales-Hurtado; Patrick Meffre; Hendrik Szurmant; Zohra Benfodda
Journal:  Med Res Rev       Date:  2019-12-05       Impact factor: 12.944

2.  Thiazolidione derivatives targeting the histidine kinase YycG are effective against both planktonic and biofilm-associated Staphylococcus epidermidis.

Authors:  Ren-zheng Huang; Li-kang Zheng; Hua-yong Liu; Bin Pan; Jian Hu; Tao Zhu; Wei Wang; Dan-bin Jiang; Yang Wu; You-cong Wu; Shi-qing Han; Di Qu
Journal:  Acta Pharmacol Sin       Date:  2012-01-09       Impact factor: 6.150

3.  Efficacy of novel antibacterial compounds targeting histidine kinase YycG protein.

Authors:  Huayong Liu; Dan Zhao; Jun Chang; Liang Yan; Fuju Zhao; Youcong Wu; Tao Xu; Ting Gong; Li Chen; Nianan He; Yang Wu; Shiqing Han; Di Qu
Journal:  Appl Microbiol Biotechnol       Date:  2014-04-17       Impact factor: 4.813

Review 4.  Skin whitening agents: medicinal chemistry perspective of tyrosinase inhibitors.

Authors:  Thanigaimalai Pillaiyar; Manoj Manickam; Vigneshwaran Namasivayam
Journal:  J Enzyme Inhib Med Chem       Date:  2017-12       Impact factor: 5.051

5.  Efficient Synthesis of Novel Pyridine-Based Derivatives via Suzuki Cross-Coupling Reaction of Commercially Available 5-Bromo-2-methylpyridin-3-amine: Quantum Mechanical Investigations and Biological Activities.

Authors:  Gulraiz Ahmad; Nasir Rasool; Hafiz Mansoor Ikram; Samreen Gul Khan; Tariq Mahmood; Khurshid Ayub; Muhammad Zubair; Eman Al-Zahrani; Usman Ali Rana; Muhammad Nadeem Akhtar; Noorjahan Banu Alitheen
Journal:  Molecules       Date:  2017-01-27       Impact factor: 4.411

Review 6.  Recent Advances in Histidine Kinase-Targeted Antimicrobial Agents.

Authors:  Hongtong Chen; Chengqi Yu; Han Wu; Guoqing Li; Congran Li; Wei Hong; Xinyi Yang; Hao Wang; Xuefu You
Journal:  Front Chem       Date:  2022-07-04       Impact factor: 5.545
  6 in total

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