Literature DB >> 20264585

Tetrahydroacridones and related compounds as antimalarials.

J M L STEPHEN, I M TONKIN, J WALKER.   

Abstract

Entities:  

Keywords:  ANTIMALARIAL/tetrahydroacridone; TETRAHYDROACRIDONE/antimalarial

Mesh：

Substances：

Year:  1947        PMID： 20264585     DOI： 10.1039/jr9470001034

Source DB:  PubMed          Journal:  J Chem Soc        ISSN： 0368-1769


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  9 in total

1.  Synthesis and structure-activity relationships of antimalarial 4-oxo-3-carboxyl quinolones.

Authors:  Yiqun Zhang; W Armand Guiguemde; Martina Sigal; Fangyi Zhu; Michele C Connelly; Solomon Nwaka; R Kiplin Guy
Journal:  Bioorg Med Chem       Date:  2010-02-11       Impact factor: 3.641

2.  4(1H)-pyridone and 4(1H)-quinolone derivatives as antimalarials with erythrocytic, exoerythrocytic, and transmission blocking activities.

Authors:  Andrii Monastyrskyi; Dennis E Kyle; Roman Manetsch
Journal:  Curr Top Med Chem       Date:  2014       Impact factor: 3.295

3.  Lead optimization of 3-carboxyl-4(1H)-quinolones to deliver orally bioavailable antimalarials.

Authors:  Yiqun Zhang; Julie A Clark; Michele C Connelly; Fangyi Zhu; Jaeki Min; W Armand Guiguemde; Anupam Pradhan; Lalitha Iyer; Anna Furimsky; Jason Gow; Toufan Parman; Farah El Mazouni; Margaret A Phillips; Dennis E Kyle; Jon Mirsalis; R Kiplin Guy
Journal:  J Med Chem       Date:  2012-04-18       Impact factor: 7.446

4.  Potent Antimalarial 2-Pyrazolyl Quinolone bc 1 (Qi) Inhibitors with Improved Drug-like Properties.

Authors:  W David Hong; Suet C Leung; Kangsa Amporndanai; Jill Davies; Richard S Priestley; Gemma L Nixon; Neil G Berry; S Samar Hasnain; Svetlana Antonyuk; Stephen A Ward; Giancarlo A Biagini; Paul M O'Neill
Journal:  ACS Med Chem Lett       Date:  2018-10-19       Impact factor: 4.345

Review 5.  Antibiotics in malaria therapy: which antibiotics except tetracyclines and macrolides may be used against malaria?

Authors:  Tiphaine Gaillard; Marylin Madamet; Francis Foguim Tsombeng; Jérôme Dormoi; Bruno Pradines
Journal:  Malar J       Date:  2016-11-15       Impact factor: 2.979

6.  Targeting the Ubiquinol-Reduction (Qi) Site of the Mitochondrial Cytochrome bc1 Complex for the Development of Next Generation Quinolone Antimalarials.

Authors:  Kangsa Amporndanai; Nattapon Pinthong; Paul M O'Neill; W David Hong; Richard K Amewu; Chandrakala Pidathala; Neil G Berry; Suet C Leung; Stephen A Ward; Giancarlo A Biagini; S Samar Hasnain; Svetlana V Antonyuk
Journal:  Biology (Basel)       Date:  2022-07-25

7.  ICI 56,780 Optimization: Structure-Activity Relationship Studies of 7-(2-Phenoxyethoxy)-4(1H)-quinolones with Antimalarial Activity.

Authors:  Jordany R Maignan; Cynthia L Lichorowic; James Giarrusso; Lynn D Blake; Debora Casandra; Tina S Mutka; Alexis N LaCrue; Jeremy N Burrows; Paul A Willis; Dennis E Kyle; Roman Manetsch
Journal:  J Med Chem       Date:  2016-07-12       Impact factor: 8.039

Review 8.  Recent progress in the development of anti-malarial quinolones.

Authors:  Richard M Beteck; Frans J Smit; Richard K Haynes; David D N'Da
Journal:  Malar J       Date:  2014-08-30       Impact factor: 2.979

9.  1,2-substituted 4-(1H)-quinolones: synthesis, antimalarial and antitrypanosomal activities in vitro.

Authors:  Abraham Wube; Antje Hüfner; Werner Seebacher; Marcel Kaiser; Reto Brun; Rudolf Bauer; Franz Bucar
Journal:  Molecules       Date:  2014-09-10       Impact factor: 4.411
  9 in total

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