Literature DB >> 20224985

Comparison of drug permeabilities and BCS classification: three lipid-component PAMPA system method versus Caco-2 monolayers.

Zeynep S Teksin1, Paul R Seo, James E Polli.   

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Year:  2010        PMID： 20224985      PMCID： PMC2844511          DOI： 10.1208/s12248-010-9176-2

Source DB:  PubMed          Journal:  AAPS J        ISSN： 1550-7416            Impact factor:   4.009


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  32 in total

1.  A comparative study of artificial membrane permeability assay for high throughput profiling of drug absorption potential.

Authors:  Chengyue Zhu; Lan Jiang; Teng-Man Chen; Kin-Kai Hwang
Journal:  Eur J Med Chem       Date:  2002-05       Impact factor: 6.514

2.  Biowaiver monographs for immediate release solid oral dosage forms based on biopharmaceutics classification system (BCS) literature data: verapamil hydrochloride, propranolol hydrochloride, and atenolol.

Authors:  H Vogelpoel; J Welink; G L Amidon; H E Junginger; K K Midha; H Möller; M Olling; V P Shah; D M Barends
Journal:  J Pharm Sci       Date:  2004-08       Impact factor: 3.534

3.  Drug absorption in vitro model: filter-immobilized artificial membranes. 2. Studies of the permeability properties of lactones in Piper methysticum Forst.

Authors:  A Avdeef; M Strafford; E Block; M P Balogh; W Chambliss; I Khan
Journal:  Eur J Pharm Sci       Date:  2001-12       Impact factor: 4.384

4.  Evaluation of using dog as an animal model to study the fraction of oral dose absorbed of 43 drugs in humans.

Authors:  W L Chiou; H Y Jeong; S M Chung; T C Wu
Journal:  Pharm Res       Date:  2000-02       Impact factor: 4.200

5.  Permeation characteristics of a hydrophilic basic compound across a bio-mimetic artificial membrane.

Authors:  Kiyohiko Sugano; Yoshiaki Nabuchi; Minoru Machida; Yoshinori Asoh
Journal:  Int J Pharm       Date:  2004-05-04       Impact factor: 5.875

6.  Transport evaluation of salicylic acid and structurally related compounds across Caco-2 cell monolayers and artificial PAMPA membranes.

Authors:  Maija Koljonen; Katja Rousu; Jakub Cierny; Ann Marie Kaukonen; Jouni Hirvonen
Journal:  Eur J Pharm Biopharm       Date:  2008-06-06       Impact factor: 5.571

7.  Permeation prediction of M100240 using the parallel artificial membrane permeability assay.

Authors:  Kin-Kai Hwang; Nancy E Martin; Lan Jiang; Chengyue Zhu
Journal:  J Pharm Pharm Sci       Date:  2003 Sep-Dec       Impact factor: 2.327

8.  Characterization of dexloxiglumide in vitro biopharmaceutical properties and active transport.

Authors:  Sanna Tolle-Sander; Andreas Grill; Hemant Joshi; Ram Kapil; Stefano Persiani; James E Polli
Journal:  J Pharm Sci       Date:  2003-10       Impact factor: 3.534

9.  PAMPA--a drug absorption in vitro model 7. Comparing rat in situ, Caco-2, and PAMPA permeability of fluoroquinolones.

Authors:  Marival Bermejo; Alex Avdeef; Ana Ruiz; Ricardo Nalda; Jeffrey A Ruell; Oksana Tsinman; Isabel González; Carlos Fernández; Gloria Sánchez; Teresa M Garrigues; Virginia Merino
Journal:  Eur J Pharm Sci       Date:  2004-03       Impact factor: 4.384

10.  Combined application of parallel artificial membrane permeability assay and Caco-2 permeability assays in drug discovery.

Authors:  Edward H Kerns; Li Di; Susan Petusky; Michele Farris; Rob Ley; Phil Jupp
Journal:  J Pharm Sci       Date:  2004-06       Impact factor: 3.534
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  10 in total

1.  Development of a Novel Maternal-Fetal Physiologically Based Pharmacokinetic Model II: Verification of the model for passive placental permeability drugs.

Authors:  Zufei Zhang; Jashvant D Unadkat
Journal:  Drug Metab Dispos       Date:  2017-01-03       Impact factor: 3.922

2.  Predicting the extent of metabolism using in vitro permeability rate measurements and in silico permeability rate predictions.

Authors:  Chelsea M Hosey; Leslie Z Benet
Journal:  Mol Pharm       Date:  2015-04-23       Impact factor: 4.939

3.  Anthranilic acid-containing cyclic tetrapeptides: at the crossroads of conformational rigidity and synthetic accessibility.

Authors:  Dongyue Xin; Kevin Burgess
Journal:  Org Biomol Chem       Date:  2016-05-13       Impact factor: 3.876

4.  Applying Biopharmaceutical Classification System (BCS) Criteria to Predict Oral Absorption of Drugs in Dogs: Challenges and Pitfalls.

Authors:  Mark G Papich; Marilyn N Martinez
Journal:  AAPS J       Date:  2015-04-29       Impact factor: 4.009

Review 5.  Physiologically based pharmacokinetic models: integration of in silico approaches with micro cell culture analogues.

Authors:  A Chen; M L Yarmush; T Maguire
Journal:  Curr Drug Metab       Date:  2012-07       Impact factor: 3.731

6.  Robotically handled whole-tissue culture system for the screening of oral drug formulations.

Authors:  Thomas von Erlach; Sarah Saxton; Yunhua Shi; Daniel Minahan; Daniel Reker; Farhad Javid; Young-Ah Lucy Lee; Carl Schoellhammer; Tina Esfandiary; Cody Cleveland; Lucas Booth; Jiaqi Lin; Hannah Levy; Sophie Blackburn; Alison Hayward; Robert Langer; Giovanni Traverso
Journal:  Nat Biomed Eng       Date:  2020-04-27       Impact factor: 25.671

7.  Functional Group Distributions, Partition Coefficients, and Resistance Factors in Lipid Bilayers Using Site Identification by Ligand Competitive Saturation.

Authors:  Christoffer Lind; Poonam Pandey; Richard W Pastor; Alexander D MacKerell
Journal:  J Chem Theory Comput       Date:  2021-04-30       Impact factor: 6.006

8.  Effect of Coformer Selection on In Vitro and In Vivo Performance of Adefovir Dipivoxil Cocrystals.

Authors:  Luyuan Li; Zunting Pang; Kun Ma; Yuan Gao; Daoyi Zheng; Yuanfeng Wei; Jianjun Zhang; Shuai Qian
Journal:  Pharm Res       Date:  2021-11-02       Impact factor: 4.200

9.  Fate of ingested Clostridium difficile spores in mice.

Authors:  Amber Howerton; Manomita Patra; Ernesto Abel-Santos
Journal:  PLoS One       Date:  2013-08-30       Impact factor: 3.240

10.  Discovery of the first N-hydroxycinnamamide-based histone deacetylase 1/3 dual inhibitors with potent oral antitumor activity.

Authors:  Xiaoyang Li; Elizabeth S Inks; Xiaoguang Li; Jinning Hou; C James Chou; Jian Zhang; Yuqi Jiang; Yingjie Zhang; Wenfang Xu
Journal:  J Med Chem       Date:  2014-04-15       Impact factor: 7.446
  10 in total

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