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10 in total

1. 2-aminothiazole-derived opioids. Bioisosteric replacement of phenols.

Authors: Ao Zhang; Wennan Xiong; James E Hilbert; Emily K DeVita; Jean M Bidlack; John L Neumeyer
Journal: J Med Chem Date: 2004-04-08 Impact factor: 7.446

2. A Hantzsch synthesis of 2-aminothiazoles performed in a heated microreactor system.

Authors: Eduardo Garcia-Egido; Stephanie Y Wong; Brian H Warrington
Journal: Lab Chip Date: 2002-01-18 Impact factor: 6.799

3. General method for the rapid solid-phase synthesis of large numbers of peptides: specificity of antigen-antibody interaction at the level of individual amino acids.

Authors: R A Houghten
Journal: Proc Natl Acad Sci U S A Date: 1985-08 Impact factor: 11.205

4. Novel structural templates for estrogen-receptor ligands and prospects for combinatorial synthesis of estrogens.

Authors: B E Fink; D S Mortensen; S R Stauffer; Z D Aron; J A Katzenellenbogen
Journal: Chem Biol Date: 1999-04

5. 3-[1-(2-Benzoxazolyl)hydrazino]propanenitrile derivatives: inhibitors of immune complex induced inflammation.

Authors: F Haviv; J D Ratajczyk; R W DeNet; F A Kerdesky; R L Walters; S P Schmidt; J H Holms; P R Young; G W Carter
Journal: J Med Chem Date: 1988-09 Impact factor: 7.446

6. Structure-activity relationships of a series of 2-amino-4-thiazole-containing renin inhibitors.

Authors: W C Patt; H W Hamilton; M D Taylor; M J Ryan; D G Taylor; C J Connolly; A M Doherty; S R Klutchko; I Sircar; B A Steinbaugh
Journal: J Med Chem Date: 1992-07-10 Impact factor: 7.446

7. Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists.

Authors: J E van Muijlwijk-Koezen; H Timmerman; R C Vollinga; J Frijtag von Drabbe Künzel; M de Groote; S Visser; A P IJzerman
Journal: J Med Chem Date: 2001-03-01 Impact factor: 7.446

8. N-(4-substituted-thiazolyl)oxamic acid derivatives, a new series of potent, orally active antiallergy agents.

Authors: K D Hargrave; F K Hess; J T Oliver
Journal: J Med Chem Date: 1983-08 Impact factor: 7.446

9. 4-Hydroxy-3-quinolinecarboxamides with antiarthritic and analgesic activities.

Authors: F Clemence; O Le Martret; F Delevallee; J Benzoni; A Jouanen; S Jouquey; M Mouren; R Deraedt
Journal: J Med Chem Date: 1988-07 Impact factor: 7.446

10. 4-(1,2,5,6-Tetrahydro-1-alkyl-3-pyridinyl)-2-thiazolamines: a novel class of compounds with central dopamine agonist properties.

Authors: J C Jaen; L D Wise; B W Caprathe; H Tecle; S Bergmeier; C C Humblet; T G Heffner; L T Meltzer; T A Pugsley
Journal: J Med Chem Date: 1990-01 Impact factor: 7.446

10 in total

3 in total

1. N-terminus 4-Chloromethyl Thiazole Peptide as a Macrocyclization Tool in the Synthesis of Cyclic Peptides: Application to the Synthesis of Conformationally Constrained RGD-Containing Integrin Ligands.

Authors: Adel Nefzi; Jason E Fenwick
Journal: Tetrahedron Lett Date: 2011-02-16 Impact factor: 2.415

2. Two-Steps Hantzsch Based Macrocyclization Approach for the Synthesis of Thiazole Containing Cyclopeptides.

Authors: Adel Nefzi; Sergey Arutyunyan; Jason E Fenwick
Journal: J Org Chem Date: 2010-11-19 Impact factor: 4.354

3. Bis-Cyclic Guanidine Heterocyclic Peptidomimetics as Opioid Ligands with Mixed μ-, κ- and δ-Opioid Receptor Interactions: A Potential Approach to Novel Analgesics.

Authors: Jay P McLaughlin; Ramanjaneyulu Rayala; Ashley J Bunnell; Mukund P Tantak; Shainnel O Eans; Khadija Nefzi; Michelle L Ganno; Colette T Dooley; Adel Nefzi
Journal: Int J Mol Sci Date: 2022-08-25 Impact factor: 6.208

3 in total