Literature DB >> 20161438

Synthesis of labeled meropenem for the analysis of M. tuberculosis transpeptidases.

David B Kastrinsky1, Clifton E Barry.   

Abstract

A concise synthesis of (14)C labeled meropenem prepared from (14)C dimethylamine hydrochloride is described. Using a similar reaction sequence, the meropenem nucleus was also attached to biotin providing a probe for protein interaction studies.

Entities:  

Year:  2010        PMID： 20161438      PMCID： PMC2789577          DOI： 10.1016/j.tetlet.2009.10.124

Source DB:  PubMed          Journal:  Tetrahedron Lett        ISSN： 0040-4039            Impact factor:   2.415


  29 in total

Review 1.  Biochemistry and comparative genomics of SxxK superfamily acyltransferases offer a clue to the mycobacterial paradox: presence of penicillin-susceptible target proteins versus lack of efficiency of penicillin as therapeutic agent.

Authors:  Colette Goffin; Jean-Marie Ghuysen
Journal:  Microbiol Mol Biol Rev       Date:  2002-12       Impact factor: 11.056

2.  Novel mechanism of resistance to glycopeptide antibiotics in Enterococcus faecium.

Authors:  Julie Cremniter; Jean-Luc Mainardi; Nathalie Josseaume; Jean-Charles Quincampoix; Lionel Dubost; Jean-Emmanuel Hugonnet; Arul Marie; Laurent Gutmann; Louis B Rice; Michel Arthur
Journal:  J Biol Chem       Date:  2006-08-29       Impact factor: 5.157

3.  The vitro efficacy of beta-lactam and beta-lactamase inhibitors against multidrug resistant clinical strains of Mycobacterium tuberculosis.

Authors:  Irem Dinçer; Alper Ergin; Tanil Kocagöz
Journal:  Int J Antimicrob Agents       Date:  2004-04       Impact factor: 5.283

Review 4.  Carbapenems: a potent class of antibiotics.

Authors:  David P Nicolau
Journal:  Expert Opin Pharmacother       Date:  2008-01       Impact factor: 3.889

5.  Balance between two transpeptidation mechanisms determines the expression of beta-lactam resistance in Enterococcus faecium.

Authors:  Jean-Luc Mainardi; Véronique Morel; Martine Fourgeaud; Julie Cremniter; Didier Blanot; Raymond Legrand; Claude Frehel; Michel Arthur; Jean Van Heijenoort; Laurent Gutmann
Journal:  J Biol Chem       Date:  2002-06-19       Impact factor: 5.157

Review 6.  Thienamycin: development of imipenen-cilastatin.

Authors:  F M Kahan; H Kropp; J G Sundelof; J Birnbaum
Journal:  J Antimicrob Chemother       Date:  1983-12       Impact factor: 5.790

Review 7.  The envelope of mycobacteria.

Authors:  P J Brennan; H Nikaido
Journal:  Annu Rev Biochem       Date:  1995       Impact factor: 23.643

Review 8.  Meropenem: a microbiological overview.

Authors:  J R Edwards
Journal:  J Antimicrob Chemother       Date:  1995-07       Impact factor: 5.790

9.  Synthesis and preliminary biological evaluation of (3-iodobenzoyl)norbiotinamide and ((5-iodo-3-pyridinyl)carbonyl)norbiotinamide: two radioiodinated biotin conjugates with improved stability.

Authors:  C F Foulon; K L Alston; M R Zalutsky
Journal:  Bioconjug Chem       Date:  1997 Mar-Apr       Impact factor: 4.774

Review 10.  Evolution of peptidoglycan biosynthesis under the selective pressure of antibiotics in Gram-positive bacteria.

Authors:  Jean-Luc Mainardi; Régis Villet; Timothy D Bugg; Claudine Mayer; Michel Arthur
Journal:  FEMS Microbiol Rev       Date:  2008-02-11       Impact factor: 16.408
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  2 in total

1.  Nonclassical transpeptidases of Mycobacterium tuberculosis alter cell size, morphology, the cytosolic matrix, protein localization, virulence, and resistance to β-lactams.

Authors:  Maia K Schoonmaker; William R Bishai; Gyanu Lamichhane
Journal:  J Bacteriol       Date:  2014-01-24       Impact factor: 3.490

Review 2.  Cell wall peptidoglycan in Mycobacterium tuberculosis: An Achilles' heel for the TB-causing pathogen.

Authors:  Arundhati Maitra; Tulika Munshi; Jess Healy; Liam T Martin; Waldemar Vollmer; Nicholas H Keep; Sanjib Bhakta
Journal:  FEMS Microbiol Rev       Date:  2019-09-01       Impact factor: 16.408
  2 in total

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