Literature DB >> 20131879

[4 + 2] Cycloaddition reactions catalyzed by a chiral oxazaborolidinium cation. Reaction rates and diastereo-, regio-, and enantioselectivity depend on whether both bonds are formed simultaneously.

Santanu Mukherjee1, E J Corey.   

Abstract

The reaction rates and products in enantioselective Diels-Alder reactions with a range of dienophiles correlate with the expected degree of concertedness of bond formation in the transition state.

Entities:  

Year:  2010        PMID： 20131879     DOI： 10.1021/ol100032u

Source DB:  PubMed          Journal:  Org Lett        ISSN： 1523-7052            Impact factor:   6.005


  5 in total

1.  Nature Inspired Molecular Design: Stereoselective Synthesis of Bicyclic and Polycyclic Ethers for Potent HIV-1 Protease Inhibitors.

Authors:  Arun K Ghosh; Margherita Brindisi
Journal:  Asian J Org Chem       Date:  2018-06-08       Impact factor: 3.319

2.  Design and Development of Highly Potent HIV-1 Protease Inhibitors with a Crown-Like Oxotricyclic Core as the P2-Ligand To Combat Multidrug-Resistant HIV Variants.

Authors:  Arun K Ghosh; Kalapala Venkateswara Rao; Prasanth R Nyalapatla; Heather L Osswald; Cuthbert D Martyr; Manabu Aoki; Hironori Hayashi; Johnson Agniswamy; Yuan-Fang Wang; Haydar Bulut; Debananda Das; Irene T Weber; Hiroaki Mitsuya
Journal:  J Med Chem       Date:  2017-04-18       Impact factor: 7.446

3.  Mechanisms and Specificity of Phenazine Biosynthesis Protein PhzF.

Authors:  Christina Diederich; Mario Leypold; Martin Culka; Hansjörg Weber; Rolf Breinbauer; G Matthias Ullmann; Wulf Blankenfeldt
Journal:  Sci Rep       Date:  2017-07-24       Impact factor: 4.379

4.  Asymmetric Diels-Alder reaction of 3-(acyloxy) acryloyl oxazolidinones: optically active synthesis of a high-affinity ligand for potent HIV-1 protease inhibitors.

Authors:  Arun K Ghosh; Alessandro Grillo; Satish Kovela; Margherita Brindisi
Journal:  RSC Adv       Date:  2019-12-17       Impact factor: 4.036

5.  Overcoming synthetic challenges in targeting coenzyme A biosynthesis with the antimicrobial natural product CJ-15,801.

Authors:  Riyad Domingo; Renier van der Westhuyzen; Anton R Hamann; Konrad J Mostert; Leanne Barnard; Tanya Paquet; Erick T Tjhin; Kevin J Saliba; Willem A L van Otterlo; Erick Strauss
Journal:  Medchemcomm       Date:  2019-10-17       Impact factor: 3.597
  5 in total

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