Literature DB >> 20046884

Clinical Perspective and Recent Development of PET Radioligands for Imaging Cerebral Nicotinic Acetylcholine Receptors.

Andrew G Horti, Dean F Wong.   

Abstract

Entities:  

Year:  2009        PMID： 20046884      PMCID： PMC2761691          DOI： 10.1016/j.cpet.2009.04.014

Source DB:  PubMed          Journal:  PET Clin        ISSN： 1556-8598


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  56 in total

1.  Chemical modification of epibatidine causes a switch from agonist to antagonist and modifies its selectivity for neuronal nicotinic acetylcholine receptors.

Authors:  J E Spang; S Bertrand; G Westera; J T Patt; P A Schubiger; D Bertrand
Journal:  Chem Biol       Date:  2000-07

2.  In vivo imaging of human cerebral nicotinic acetylcholine receptors with 2-18F-fluoro-A-85380 and PET.

Authors:  Jean-Dominique Gallezot; Michel Bottlaender; Marie-Claude Grégoire; Dimitri Roumenov; Jean-Robert Deverre; Christine Coulon; Michèle Ottaviani; Frédéric Dollé; André Syrota; Héric Valette
Journal:  J Nucl Med       Date:  2005-02       Impact factor: 10.057

3.  Simplified quantification of nicotinic receptors with 2[18F]F-A-85380 PET.

Authors:  Sascha Mitkovski; Victor L Villemagne; Kathy E Novakovic; Graeme O'Keefe; Henri Tochon-Danguy; Rachel S Mulligan; Kerryn L Dickinson; Tim Saunder; Marie-Claude Gregoire; Michel Bottlaender; Frederic Dolle; Christopher C Rowe
Journal:  Nucl Med Biol       Date:  2005-08       Impact factor: 2.408

4.  Quantification of nicotinic acetylcholine receptors in the human brain with PET: bolus plus infusion administration of 2-[18F]F-A85380.

Authors:  Alane S Kimes; Svetlana I Chefer; John A Matochik; Carlo S Contoreggi; D Bruce Vaupel; Elliot A Stein; Alexey G Mukhin
Journal:  Neuroimage       Date:  2007-09-19       Impact factor: 6.556

Review 5.  Imaging brain cholinergic activity with positron emission tomography: its role in the evaluation of cholinergic treatments in Alzheimer's dementia.

Authors:  N D Volkow; Y S Ding; J S Fowler; S J Gatley
Journal:  Biol Psychiatry       Date:  2001-02-01       Impact factor: 13.382

6.  Effect of acetylcholinesterase inhibitors on the binding of nicotinic alpha4beta2 receptor PET radiotracer, (18)F-nifene: A measure of acetylcholine competition.

Authors:  Balasubramaniam Easwaramoorthy; Rama Pichika; Daphne Collins; Steven G Potkin; Frances M Leslie; Jogeshwar Mukherjee
Journal:  Synapse       Date:  2007-01       Impact factor: 2.562

7.  6-[18F]fluoro-A-85380, a novel radioligand for in vivo imaging of central nicotinic acetylcholine receptors.

Authors:  A G Horti; S I Chefer; A G Mukhin; A O Koren; D Gündisch; J M Links; V Kurian; R F Dannals; E D London
Journal:  Life Sci       Date:  2000-06-16       Impact factor: 5.037

Review 8.  Neuronal nicotinic receptors in the human brain.

Authors:  D Paterson; A Nordberg
Journal:  Prog Neurobiol       Date:  2000-05       Impact factor: 11.685

9.  Epibatidine analogues as selective ligands for the alpha(x)beta2-containing subtypes of nicotinic acetylcholine receptors.

Authors:  Yiyun Huang; Zhihong Zhu; Yingxian Xiao; Marc Laruelle
Journal:  Bioorg Med Chem Lett       Date:  2005-10-01       Impact factor: 2.823

10.  Evaluation of 5-(2-(4-pyridinyl)vinyl)-6-chloro-3-(1-methyl-2-(S)-pyrrolidinylmethoxy)pyridine and its analogues as PET radioligands for imaging nicotinic acetylcholine receptors.

Authors:  LaVerne Brown; Svetlana Chefer; Olga Pavlova; D Bruce Vaupel; Andrei O Koren; Alane S Kimes; Andrew G Horti; Alexey G Mukhin
Journal:  J Neurochem       Date:  2004-11       Impact factor: 5.372
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  8 in total

1.  Positron emission tomography experience with 2-[¹⁸F]fluoro-3-(2(S)-azetidinylmethoxy)pyridine (2-[¹⁸F]FA) in the living human brain of smokers with paranoid schizophrenia.

Authors:  James Robert Brašić; Nicola Cascella; Anil Kumar; Yun Zhou; John Hilton; Vanessa Raymont; Andrew Crabb; Maria Rita Guevara; Andrew G Horti; Dean Foster Wong
Journal:  Synapse       Date:  2011-12-29       Impact factor: 2.562

2.  Synthesis and evaluation of new radioligands [(11)C]A-833834 and [(11)C]A-752274 for positron-emission tomography of α7-nicotinic acetylcholine receptors.

Authors:  Andrew G Horti; Hayden T Ravert; Yongjun Gao; Daniel P Holt; William H Bunnelle; Michael R Schrimpf; Tao Li; Jianguo Ji; Heather Valentine; Ursula Scheffel; Hiroto Kuwabara; Dean F Wong; Robert F Dannals
Journal:  Nucl Med Biol       Date:  2013-01-05       Impact factor: 2.408

Review 3.  Imaging radiation-induced normal tissue injury.

Authors:  Mike E Robbins; Judy K Brunso-Bechtold; Ann M Peiffer; Christina I Tsien; Janet E Bailey; Lawrence B Marks
Journal:  Radiat Res       Date:  2012-02-21       Impact factor: 2.841

4.  5-(5-(6-[(11)C]methyl-3,6-diazabicyclo[3.2.0]heptan-3-yl)pyridin-2-yl)-1H-indole as a potential PET radioligand for imaging cerebral α7-nAChR in mice.

Authors:  Yongjun Gao; Hayden T Ravert; Heather Valentine; Ursula Scheffel; Paige Finley; Dean F Wong; Robert F Dannals; Andrew G Horti
Journal:  Bioorg Med Chem       Date:  2012-05-04       Impact factor: 3.641

5.  18F-XTRA PET for Enhanced Imaging of the Extrathalamic α4β2 Nicotinic Acetylcholine Receptor.

Authors:  Jennifer M Coughlin; Stephanie Slania; Yong Du; Hailey B Rosenthal; Wojciech G Lesniak; Il Minn; Gwenn S Smith; Robert F Dannals; Hiroto Kuwabara; Dean F Wong; Yuchuan Wang; Andrew G Horti; Martin G Pomper
Journal:  J Nucl Med       Date:  2018-03-01       Impact factor: 10.057

6.  Imaging α4β2 Nicotinic Acetylcholine Receptors (nAChRs) in Baboons with [18F]XTRA, a Radioligand with Improved Specific Binding in Extra-Thalamic Regions.

Authors:  Hiroto Kuwabara; Yongjun Gao; Michael Stabin; Jennifer Coughlin; Sridhar Nimmagadda; Robert F Dannals; Martin G Pomper; Andrew G Horti
Journal:  Mol Imaging Biol       Date:  2017-04       Impact factor: 3.488

Review 7.  Development of [(18)F]ASEM, a specific radiotracer for quantification of the α7-nAChR with positron-emission tomography.

Authors:  Andrew G Horti
Journal:  Biochem Pharmacol       Date:  2015-07-29       Impact factor: 5.858

Review 8.  Imaging in sepsis-associated encephalopathy--insights and opportunities.

Authors:  Daniel J Stubbs; Adam K Yamamoto; David K Menon
Journal:  Nat Rev Neurol       Date:  2013-09-03       Impact factor: 42.937
  8 in total

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