Literature DB >> 20041339

A phase I study of S-1 treatment with a 3 week schedule in advanced biliary cancer patients with or without hepatic dysfunction.

Dok Hyun Yoon1, Hyo Jung Lee, Yong Sang Hong, Kyu-Pyo Kim, Sung Sook Lee, Jae-Lyun Lee, Heung Moon Chang, Min-Hee Ryu, Yoon-Koo Kang, Jung Shin Lee, Tae Won Kim.   

Abstract

PURPOSE: A 3 week treatment schedule consisting of 2 weeks of S-1 therapy and 1 week of no therapy was introduced to reduce the toxicity and increase the convenience of combination chemotherapy. Hepatic dysfunction (HD) is common in patients with biliary tract cancer. A phase I study was conducted to assess the effects of a 3 week treatment schedule in Asian patients with or without HD.
METHODS: Forty-six patients were stratified into four groups, according to the HD criteria of the National Cancer Institute Organ Dysfunction Working Group. A three dose escalation schema was used.
RESULTS: In the normal hepatic function group, two dose-limiting toxicity (DLT) events occurred among 12 patients at the prespecified maximal dose of 100 mg/m²/day. This dose was thereby established as the maximal tolerable dose (MTD). No DLT events were observed at the predefined maximal dose of 80 mg/m²/day in the mild HD group. In the moderate HD group, two DLT events occurred among five patients treated with 80 mg/m²/day, and the MTD was defined as 70 mg/m²/day. Two of six subjects in the severe HD group experienced DLT events at doses of 60 mg/m²/day and none developed DLT events at 50 mg/m²/day.
CONCLUSIONS: The MTDs for a 3 week schedule of S-1 treatment were defined in patients with or without hepatic dysfunction. A 3 week treatment regimen of S-1 might be a platform for combination with newer cytotoxic agents or biologics.

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Year:  2009        PMID: 20041339     DOI: 10.1007/s10637-009-9378-6

Source DB:  PubMed          Journal:  Invest New Drugs        ISSN: 0167-6997            Impact factor:   3.850


  31 in total

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4.  Phase I and pharmacokinetic study of S-1 administered for 14 days in a 21-day cycle in patients with advanced upper gastrointestinal cancer.

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6.  Phase I/II study of 3-week combination of S-1 and cisplatin chemotherapy for metastatic or recurrent gastric cancer.

Authors:  Jae-Lyun Lee; Hye Jin Kang; Yoon-Koo Kang; Min-Hee Ryu; Heung Moon Chang; Tae-Won Kim; Hee Jung Sohn; Hawk Kim; Jung Shin Lee
Journal:  Cancer Chemother Pharmacol       Date:  2007-06-20       Impact factor: 3.333

7.  CYP2A6 and the plasma level of 5-chloro-2, 4-dihydroxypyridine are determinants of the pharmacokinetic variability of tegafur and 5-fluorouracil, respectively, in Japanese patients with cancer given S-1.

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Journal:  Cancer Sci       Date:  2008-05       Impact factor: 6.716

8.  Cholangiocarcinoma. A spectrum of intrahepatic, perihilar, and distal tumors.

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9.  Effective treatment of advanced biliary tract carcinoma using 5-fluorouracil continuous infusion with cisplatin.

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Journal:  Ann Oncol       Date:  1998-06       Impact factor: 32.976

10.  Phase II study of S-1, a novel oral fluorophyrimidine derivative, in patients with metastatic colorectal carcinoma. S-1 Cooperative Colorectal Carcinoma Study Group.

Authors:  A Ohtsu; H Baba; Y Sakata; Y Mitachi; N Horikoshi; K Sugimachi; T Taguchi
Journal:  Br J Cancer       Date:  2000-07       Impact factor: 7.640

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