Literature DB >> 20036039

Synthesis, in vitro antibacterial and antifungal evaluations of new alpha-hydroxyphosphonate and new alpha-acetoxyphosphonate derivatives of tetrazolo [1, 5-a] quinoline.

Amol H Kategaonkar1, Rajkumar U Pokalwar, Swapnil S Sonar, Vaibhav U Gawali, Bapurao B Shingate, Murlidhar S Shingare.   

Abstract

A series of new alpha-hydroxyphosphonate and alpha-acetoxyphosphonate derivatives have been synthesized for the first time of tetrazolo [1, 5-a] quinoline derivatives. Elemental analysis, IR, (1)H NMR, (13)C NMR and mass spectral data elucidated the structures of the all newly synthesized compounds. In vitro antimicrobial activities of the synthesized compounds were investigated against Gram-positive Bacillus subtilis, Gram-negative Escherichia coli and fungi Candida albicans and Aspergillus niger. Some of the tested compounds showed significant antimicrobial activity. Copyright (c) 2009 Elsevier Masson SAS. All rights reserved.

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Year:  2009        PMID: 20036039     DOI: 10.1016/j.ejmech.2009.12.013

Source DB:  PubMed          Journal:  Eur J Med Chem        ISSN: 0223-5234            Impact factor:   6.514


  14 in total

1.  Electrospray ionization mass spectrometry of palladium(II) quinolinylaminophosphonate complexes.

Authors:  Marina Juribašić; Lisa Bellotto; Pietro Traldi; Ljerka Tušek-Božić
Journal:  J Am Soc Mass Spectrom       Date:  2011-07-12       Impact factor: 3.109

2.  Organocatalytic High Enantioselective Synthesis of β-Formyl-α-hydroxyphosphonates.

Authors:  Sandun Perera; Vijaya Kumar Naganaboina; Long Wang; Bin Zhang; Qunsheng Guo; Laxmidhar Rout; Cong-Gui Zhao
Journal:  Adv Synth Catal       Date:  2011-06-30       Impact factor: 5.837

3.  Developing novel organocatalyzed aldol reactions for the enantioselective synthesis of biologically active molecules.

Authors:  Mayur Bhanushali; Cong-Gui Zhao
Journal:  Synthesis (Stuttg)       Date:  2011-06       Impact factor: 3.157

4.  Antigiardial activity of novel triazolyl-quinolone-based chalcone derivatives: when oxygen makes the difference.

Authors:  Vijay Bahadur; Daniela Mastronicola; Amit K Singh; Hemandra K Tiwari; Leopoldo P Pucillo; Paolo Sarti; Brajendra K Singh; Alessandro Giuffrè
Journal:  Front Microbiol       Date:  2015-04-08       Impact factor: 5.640

5.  Evaluation of fluorescence in situ hybridisation (FISH) for the detection of fungi directly from blood cultures and cerebrospinal fluid from patients with suspected invasive mycoses.

Authors:  Roberto Moreira Da Silva; João Ricardo Da Silva Neto; Carla Silvana Santos; Hagen Frickmann; Sven Poppert; Kátia Santana Cruz; Daniela Koshikene; João Vicente Braga De Souza
Journal:  Ann Clin Microbiol Antimicrob       Date:  2015-01-31       Impact factor: 3.944

6.  An oral quinoline derivative, MPT0B392, causes leukemic cells mitotic arrest and overcomes drug resistant cancer cells.

Authors:  Min-Wu Chao; Han-Li Huang; Wei-Chun HuangFu; Kai-Cheng Hsu; Yi-Min Liu; Yi-Wen Wu; Chao-Feng Lin; Yi-Lin Chen; Mei-Jung Lai; Hsueh-Yun Lee; Jing-Ping Liou; Che-Ming Teng; Chia-Ron Yang
Journal:  Oncotarget       Date:  2017-04-25

Review 7.  Synthesis and Reactions of α-Hydroxyphosphonates.

Authors:  Zita Rádai; György Keglevich
Journal:  Molecules       Date:  2018-06-20       Impact factor: 4.411

8.  Syntheses and Reactions of Pyrroline, Piperidine Nitroxide Phosphonates.

Authors:  Mostafa Isbera; Balázs Bognár; József Jekő; Cecilia Sár; Kálmán Hideg; Tamás Kálai
Journal:  Molecules       Date:  2020-05-22       Impact factor: 4.411

9.  Solvent- and Catalyst-Free One-Pot Green Bound-Type Fused Bis-Heterocycles Synthesis via Groebke-Blackburn-Bienaymé Reaction/SNAr/Ring-Chain Azido-Tautomerization Strategy.

Authors:  Miguel Ángel Claudio-Catalán; Shrikant G Pharande; Andrea Quezada-Soto; Kranthi G Kishore; Angel Rentería-Gómez; Felipe Padilla-Vaca; Rocío Gámez-Montaño
Journal:  ACS Omega       Date:  2018-05-14

10.  Antifungal activity of synthetic naphthoquinones against dermatophytes and opportunistic fungi: preliminary mechanism-of-action tests.

Authors:  Maria do Perpetuo Socorro Borges Carriço Ferreira; Mariana Filomena do Carmo Cardoso; Fernando de Carvalho da Silva; Vitor Francisco Ferreira; Emerson Silva Lima; João Vicente Braga Souza
Journal:  Ann Clin Microbiol Antimicrob       Date:  2014-07-06       Impact factor: 3.944

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