Literature DB >> 20020315

UR-60427, a novel H4 receptor-inverse agonist that shows good efficacy in a rat asthma model.

J Alfón1, N Ardanaz, B Gil-Torregrosa, A Fernández, D Balsa, E Carceller, Ll Gómez, M Merlos, J Cortijo, E Morcillo, X Bartrolí.   

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Year:  2010        PMID： 20020315     DOI： 10.1007/s00011-009-0128-1

Source DB:  PubMed          Journal:  Inflamm Res        ISSN： 1023-3830            Impact factor:   4.575


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  4 in total

Review 1.  The role of histamine H4 receptor in immune and inflammatory disorders.

Authors:  E Zampeli; E Tiligada
Journal:  Br J Pharmacol       Date:  2009-03-20       Impact factor: 8.739

2.  The histamine H4 receptor mediates allergic airway inflammation by regulating the activation of CD4+ T cells.

Authors:  Paul J Dunford; Niall O'Donnell; Jason P Riley; Kacy N Williams; Lars Karlsson; Robin L Thurmond
Journal:  J Immunol       Date:  2006-06-01       Impact factor: 5.422

3.  Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.

Authors:  Herman D Lim; Richard M van Rijn; Ping Ling; Remko A Bakker; Robin L Thurmond; Rob Leurs
Journal:  J Pharmacol Exp Ther       Date:  2005-06-09       Impact factor: 4.030

4.  A potent and selective histamine H4 receptor antagonist with anti-inflammatory properties.

Authors:  Robin L Thurmond; Pragnya J Desai; Paul J Dunford; Wai-Ping Fung-Leung; Claudia L Hofstra; Wen Jiang; Steven Nguyen; Jason P Riley; Siquan Sun; Kacy N Williams; James P Edwards; Lars Karlsson
Journal:  J Pharmacol Exp Ther       Date:  2004-01-13       Impact factor: 4.030
  4 in total

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