Literature DB >> 20001563

Optimal tolerability of ultra-low-dose continuous combined 17beta-estradiol and norethisterone acetate: laboratory and safety results.

G Samsioe1, J Hruska.   

Abstract

OBJECTIVE: To evaluate the influence of two ultra-low doses of oral continuous combined hormone therapy and placebo on metabolic parameters, and to assess safety endpoints and overall tolerability in healthy postmenopausal women.
DESIGN: In a subpopulation of the Clinical study on Hormone dose Optimisation In Climacteric symptoms Evaluation (CHOICE) trial, lipids and parameters of glucose metabolism and hemostasis were analyzed in Nordic women (n = 158) at baseline and after 12 and 24 weeks of treatment with 0.5 mg 17beta-estradiol (E2) + 0.25 mg norethisterone acetate (NETA), 0.5 mg E2 + 0.1 mg NETA or placebo. Adverse events occurring from the first trial-related activity, whether related or not related to the study medication, were recorded for the entire population (n = 575) of the trial. The seriousness, relationship to treatment and the reason for withdrawal were reported.
RESULTS: Both ultra-low-dose combinations were neutral to changes in lipid and lipoprotein, hemostasis parameters and carbohydrate metabolism during the trial. The incidence of serious adverse events was only 1% in respective treatment groups. Adverse events were the reason for withdrawal in only 2% and 6% of women in the 0.5 mg E2 + 0.25 mg and 0.1 mg NETA groups, and in 8% in the placebo group. No weight gain or change in blood pressure was reported during the trial in any of the study groups.
CONCLUSION: The treatments had neutral effects on metabolic parameters in the study population. Excellent tolerability of both ultra-low doses resulted in high completion rates.

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Year:  2010        PMID: 20001563     DOI: 10.3109/13697130903480706

Source DB:  PubMed          Journal:  Climacteric        ISSN: 1369-7137            Impact factor:   3.005


  3 in total

Review 1.  Cognitive Changes with Reproductive Aging, Perimenopause, and Menopause.

Authors:  Kelly N Morgan; Carol A Derby; Carey E Gleason
Journal:  Obstet Gynecol Clin North Am       Date:  2018-10-25       Impact factor: 2.844

2.  Effects of Hormone Therapy on Cognition and Mood in Recently Postmenopausal Women: Findings from the Randomized, Controlled KEEPS-Cognitive and Affective Study.

Authors:  Carey E Gleason; N Maritza Dowling; Whitney Wharton; JoAnn E Manson; Virginia M Miller; Craig S Atwood; Eliot A Brinton; Marcelle I Cedars; Rogerio A Lobo; George R Merriam; Genevieve Neal-Perry; Nanette F Santoro; Hugh S Taylor; Dennis M Black; Matthew J Budoff; Howard N Hodis; Frederick Naftolin; S Mitchell Harman; Sanjay Asthana
Journal:  PLoS Med       Date:  2015-06-02       Impact factor: 11.069

3.  Effects of ultra-low dose hormone therapy on biochemical bone turnover markers in postmenopausal women: A randomized, placebo-controlled, double-blind trial.

Authors:  Lucia Costa-Paiva; Maria Celeste O Wender; Rogerio B Machado; Luciano M Pompei; Eliana A Nahas; Jorge Nahas-Neto; Sonia Y Del Debbio; Mariangela Badalotti; Achilles M Cruz
Journal:  Post Reprod Health       Date:  2022-08-07
  3 in total

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