Literature DB >> 20000419

Recent advances in the discovery of competitive protein tyrosine phosphatase 1B inhibitors for the treatment of diabetes, obesity, and cancer.

Andrew P Combs1.   

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Year:  2010        PMID： 20000419     DOI： 10.1021/jm901090b

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  62 in total

1.  High-resolution dose-response screening using droplet-based microfluidics.

Authors:  Oliver J Miller; Abdeslam El Harrak; Thomas Mangeat; Jean-Christophe Baret; Lucas Frenz; Bachir El Debs; Estelle Mayot; Michael L Samuels; Eamonn K Rooney; Pierre Dieu; Martin Galvan; Darren R Link; Andrew D Griffiths
Journal:  Proc Natl Acad Sci U S A       Date:  2011-12-27       Impact factor: 11.205

2.  Protein tyrosine phosphatase 1B inhibitory activity of Indonesian herbal medicines and constituents of Cinnamomum burmannii and Zingiber aromaticum.

Authors:  Azis Saifudin; Shigetoshi Kadota; Yasuhiro Tezuka
Journal:  J Nat Med       Date:  2012-05-30       Impact factor: 2.343

3.  Regio- and Enantioselective Bromocyclization of Difluoroalkenes as a Strategy to Access Tetrasubstituted Difluoromethylene-Containing Stereocenters.

Authors:  Edward Miller; Suhong Kim; Katarina Gibson; Jeffrey S Derrick; F Dean Toste
Journal:  J Am Chem Soc       Date:  2020-04-30       Impact factor: 15.419

4.  Protein tyrosine phosphatase 1B inhibitory activities of ursane- and lupane-type triterpenes from Sorbus pohuashanensis.

Authors:  Dongxia Li; Wei Li; Koji Higai; Kazuo Koike
Journal:  J Nat Med       Date:  2013-10-06       Impact factor: 2.343

5.  The chemistry and pharmacology of privileged pyrroloquinazolines.

Authors:  Bo Chao; Bingbing X Li; Xiangshu Xiao
Journal:  Medchemcomm       Date:  2015-04-01       Impact factor: 3.597

Review 6.  Small molecule tools for functional interrogation of protein tyrosine phosphatases.

Authors:  Rongjun He; Li-Fan Zeng; Yantao He; Sheng Zhang; Zhong-Yin Zhang
Journal:  FEBS J       Date:  2012-08-16       Impact factor: 5.542

7.  Antidiabetic activity in vitro and in vivo of BDB, a selective inhibitor of protein tyrosine phosphatase 1B, from Rhodomela confervoides.

Authors:  Jiao Luo; Meiling Zheng; Bo Jiang; Chao Li; Shuju Guo; Lijun Wang; Xiangqian Li; Rilei Yu; Dayong Shi
Journal:  Br J Pharmacol       Date:  2020-08-30       Impact factor: 8.739

8.  Internal Structure and Preferential Protein Binding of Colloidal Aggregates.

Authors:  Da Duan; Hayarpi Torosyan; Daniel Elnatan; Christopher K McLaughlin; Jennifer Logie; Molly S Shoichet; David A Agard; Brian K Shoichet
Journal:  ACS Chem Biol       Date:  2016-12-16       Impact factor: 5.100

9.  Identification of Bidentate Salicylic Acid Inhibitors of PTP1B.

Authors:  Sina Haftchenary; Andriana O Jouk; Isabelle Aubry; Andrew M Lewis; Melissa Landry; Daniel P Ball; Andrew E Shouksmith; Catherine V Collins; Michel L Tremblay; Patrick T Gunning
Journal:  ACS Med Chem Lett       Date:  2015-07-22       Impact factor: 4.345

10.  Organocatalytic multicomponent reaction for the acquisition of a selective inhibitor of mPTPB, a virulence factor of tuberculosis.

Authors:  Rongjun He; Li-Fan Zeng; Yantao He; Li Wu; Andrea Michelle Gunawan; Zhong-Yin Zhang
Journal:  Chem Commun (Camb)       Date:  2013-03-11       Impact factor: 6.222
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