Literature DB >> 19954276

Vigabatrin: a comprehensive review of drug properties including clinical updates following recent FDA approval.

Justin A Tolman1, Michele A Faulkner.   

Abstract

BACKGROUND: Vigabatrin (Sabril) was approved in the USA in mid-2009 for the adjunctive treatment of refractory complex partial seizures and as treatment of infantile spasms. Vigabatrin's more than 30-year history of research and development is condensed into a clinically relevant review pertaining to this 2009 approval. METHODS/DISCUSSION: A review of the scientific literature was conducted with special focus given to the drug molecule, its mechanism of action, its effects on living systems (e.g., pharmacokinetic, pharmacologic and toxicologic), and its anticipated role among antiepileptic drugs in the USA.
CONCLUSIONS: The recent approval of vigabatrin makes a significant addition to antiepileptic drug options. The FDA implemented a Risk Evaluation and Mitigation Strategy to control for the possibility of severe adverse drug events.

Entities:  

Mesh:

Substances:

Year:  2009        PMID: 19954276     DOI: 10.1517/14656560903451690

Source DB:  PubMed          Journal:  Expert Opin Pharmacother        ISSN: 1465-6566            Impact factor:   3.889


  11 in total

1.  GAD1 Upregulation Programs Aggressive Features of Cancer Cell Metabolism in the Brain Metastatic Microenvironment.

Authors:  Patricia M Schnepp; Dennis D Lee; Ian H Guldner; Treasa K O'Tighearnaigh; Erin N Howe; Bhavana Palakurthi; Kaitlyn E Eckert; Tiffany A Toni; Brandon L Ashfeld; Siyuan Zhang
Journal:  Cancer Res       Date:  2017-04-11       Impact factor: 12.701

2.  Challenges of simultaneous measurements of brain extracellular GABA and glutamate in vivo using enzyme-coated microelectrode arrays.

Authors:  Jason J Burmeister; David A Price; François Pomerleau; Peter Huettl; Jorge E Quintero; Greg A Gerhardt
Journal:  J Neurosci Methods       Date:  2019-10-07       Impact factor: 2.390

3.  Validation of the rat model of cryptogenic infantile spasms.

Authors:  Tamar Chachua; Mi-Sun Yum; Jana Velíšková; Libor Velíšek
Journal:  Epilepsia       Date:  2011-08-19       Impact factor: 5.864

4.  CPP-115, a vigabatrin analogue, decreases spasms in the multiple-hit rat model of infantile spasms.

Authors:  Stephen W Briggs; Wenzhu Mowrey; Charles B Hall; Aristea S Galanopoulou
Journal:  Epilepsia       Date:  2013-10-28       Impact factor: 5.864

5.  Population pharmacokinetics analysis of vigabatrin in adults and children with epilepsy and children with infantile spasms.

Authors:  Jace C Nielsen; Kenneth G Kowalski; Aziz Karim; Mahlaqa Patel; David L Wesche; Dwain Tolbert
Journal:  Clin Pharmacokinet       Date:  2014-11       Impact factor: 6.447

6.  A covalent small molecule inhibitor of glutamate-oxaloacetate transaminase 1 impairs pancreatic cancer growth.

Authors:  Tomohiro Yoshida; Shingo Yamasaki; Osamu Kaneko; Naofumi Taoka; Yusuke Tomimoto; Ichiji Namatame; Toshiko Yahata; Sadao Kuromitsu; Lewis C Cantley; Costas A Lyssiotis
Journal:  Biochem Biophys Res Commun       Date:  2019-11-28       Impact factor: 3.575

7.  Probing the steric requirements of the γ-aminobutyric acid aminotransferase active site with fluorinated analogues of vigabatrin.

Authors:  Jose I Juncosa; Andrew P Groves; Guoyao Xia; Richard B Silverman
Journal:  Bioorg Med Chem       Date:  2012-12-20       Impact factor: 3.641

Review 8.  Vigabatrin versus carbamazepine monotherapy for epilepsy.

Authors:  Yousheng Xiao; Lu Gan; Jin Wang; Man Luo; Hongye Luo
Journal:  Cochrane Database Syst Rev       Date:  2015-11-18

Review 9.  Rational approaches for the design of various GABA modulators and their clinical progression.

Authors:  Kavita Bhagat; Jatinder V Singh; Piyusha P Pagare; Nitish Kumar; Anchal Sharma; Gurinder Kaur; Nihar Kinarivala; Srinivasa Gandu; Harbinder Singh; Sahil Sharma; Preet Mohinder S Bedi
Journal:  Mol Divers       Date:  2020-03-13       Impact factor: 2.943

10.  Does the Swedish Interactive Threshold Algorithm (SITA) accurately map visual field loss attributed to vigabatrin?

Authors:  Miriam L Conway; Sarah L Hosking; Haogang Zhu; Robert P Cubbidge
Journal:  BMC Ophthalmol       Date:  2014-12-23       Impact factor: 2.209

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.