Literature DB >> 19926175

Molecular iodine promoted synthesis of new pyrazolo[3,4-d]pyrimidine derivatives as potential antibacterial agents.

Mehdi Bakavoli1, Ghodsieh Bagherzadeh, Maryam Vaseghifar, Ali Shiri, Mehdi Pordel, Mansour Mashreghi, Parvaneh Pordeli, Maryam Araghi.   

Abstract

Iodocyclization of 5-amino-1-(2,4-dinitrophenyl)-1H-4-pyrazolcarboxamides with aromatic aldehydes gave a new series of pyrazolo[3,4-d]pyrimidine derivatives in a single step and their antibacterial activity comparable to Streptomycin as reference drug was evaluated. Copyright 2009 Elsevier Masson SAS. All rights reserved.

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Year:  2009        PMID： 19926175     DOI： 10.1016/j.ejmech.2009.10.051

Source DB:  PubMed          Journal:  Eur J Med Chem        ISSN： 0223-5234            Impact factor:   6.514


  11 in total

1.  Synthesis and pharmacological evaluation of pyrazolopyrimidopyrimidine derivatives: anti-inflammatory agents with gastroprotective effect in rats.

Authors:  Amine Karoui; Fatma Allouche; Monia Deghrigue; Asma Agrebi; Abderrahman Bouraoui; Fakher Chabchoub
Journal:  Med Chem Res       Date:  2013-09-04       Impact factor: 1.965

2.  Dimroth rearrangement-based synthesis of novel derivatives of [1,3]selenazolo[5,4-e][1,2,4]triazolo[1,5-c]pyrimidine as a new class of selenium-containing heterocyclic architecture.

Authors:  Seddigheh Sheikhi-Mohammareh; Ali Shiri; Joel Mague
Journal:  Mol Divers       Date:  2021-03-15       Impact factor: 2.943

3.  Design and Synthesis of New Substituted Pyrazolopyridines with Potent Antiproliferative Activity.

Authors:  Vassiliki Giannouli; Nikolaos Lougiakis; Ioannis K Kostakis; Nicole Pouli; Panagiotis Marakos; Alexios-Leandros Skaltsounis; David A Horne; Sangkil Nam; Katerina Gioti; Roxane Tenta
Journal:  Med Chem       Date:  2020       Impact factor: 2.329

Review 4.  5-Aminopyrazole as precursor in design and synthesis of fused pyrazoloazines.

Authors:  Ranjana Aggarwal; Suresh Kumar
Journal:  Beilstein J Org Chem       Date:  2018-01-25       Impact factor: 2.883

5.  Continuous-flow retro-Diels-Alder reaction: an efficient method for the preparation of pyrimidinone derivatives.

Authors:  Imane Nekkaa; Márta Palkó; István M Mándity; Ferenc Fülöp
Journal:  Beilstein J Org Chem       Date:  2018-02-01       Impact factor: 2.883

6.  Synthesis and anticancer evaluation of some novel pyrimido[5,4-e][1,2,4]triazines and pyrazolo[3,4-d]pyrimidine using DMF-DMA as methylating and cyclizing agent.

Authors:  Samar A El-Kalyoubi
Journal:  Chem Cent J       Date:  2018-05-23       Impact factor: 4.215

7.  One-Flask Synthesis of Pyrazolo[3,4-d]pyrimidines from 5-Aminopyrazoles and Mechanistic Study.

Authors:  Wan-Ping Yen; Shuo-En Tsai; Naoto Uramaru; Hiroyuki Takayama; Fung Fuh Wong
Journal:  Molecules       Date:  2017-05-16       Impact factor: 4.411

8.  Sulphonated graphene oxide catalyzed continuous flow synthesis of pyrazolo pyrimidinones, sildenafil and other PDE-5 inhibitors.

Authors:  Vinay Kumar Sthalam; Bhushan Mahajan; Purushotham Reddy Karra; Ajay K Singh; Srihari Pabbaraja
Journal:  RSC Adv       Date:  2021-12-21       Impact factor: 3.361

Review 9.  Advances in the chemical and biological diversity of heterocyclic systems incorporating pyrimido[1,6-a]pyrimidine and pyrimido[1,6-c]pyrimidine scaffolds.

Authors:  Khaled M Elattar; Başak Doğru Mert; M Monier; Ahmed El-Mekabaty
Journal:  RSC Adv       Date:  2020-04-20       Impact factor: 4.036

10.  Synthesis and Antibacterial Evaluation of New Pyrazolo[3,4-d]pyrimidines Kinase Inhibitors.

Authors:  Chiara Greco; Rosa Catania; Dario Leonardo Balacco; Vincenzo Taresco; Francesca Musumeci; Cameron Alexander; Alan Huett; Silvia Schenone
Journal:  Molecules       Date:  2020-11-16       Impact factor: 4.411
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