Literature DB >> 19904799

Evaluation of novel epothilone analogues by means of a common pharmacophore and a QSAR pseudoreceptor model for taxanes and epothilones.

Stefano Forli1, Fabrizio Manetti, Karl-Heinz Altmann, Maurizio Botta.   

Abstract

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Year:  2010        PMID： 19904799     DOI： 10.1002/cmdc.200900303

Source DB:  PubMed          Journal:  ChemMedChem        ISSN： 1860-7179            Impact factor:   3.466


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  8 in total

Review 1.  Drug discovery targeting cell division proteins, microtubules and FtsZ.

Authors:  Iwao Ojima; Kunal Kumar; Divya Awasthi; Jacob G Vineberg
Journal:  Bioorg Med Chem       Date:  2014-03-05       Impact factor: 3.641

2.  Higher sensitivity to patupilone versus paclitaxel chemotherapy in primary uterine serous papillary carcinoma cell lines with high versus low HER-2/neu expression in vitro.

Authors:  Daniel Paik; Emiliano Cocco; Stefania Bellone; Francesca Casagrande; Marta Bellone; Eric E Siegel; Christine E Richter; Peter E Schwartz; Thomas J Rutherford; Alessandro D Santin
Journal:  Gynecol Oncol       Date:  2010-07-31       Impact factor: 5.482

Review 3.  Microtubule stabilizing agents as potential treatment for Alzheimer's disease and related neurodegenerative tauopathies.

Authors:  Carlo Ballatore; Kurt R Brunden; Donna M Huryn; John Q Trojanowski; Virginia M-Y Lee; Amos B Smith
Journal:  J Med Chem       Date:  2012-09-28       Impact factor: 7.446

Review 4.  Epothilones: From discovery to clinical trials.

Authors:  Stefano Forli
Journal:  Curr Top Med Chem       Date:  2014       Impact factor: 3.295

5.  Understanding the basis of drug resistance of the mutants of αβ-tubulin dimer via molecular dynamics simulations.

Authors:  Kathiresan Natarajan; Sanjib Senapati
Journal:  PLoS One       Date:  2012-08-07       Impact factor: 3.240

6.  Synthesis and Biological Evaluation of 7-Deoxy-Epothilone Analogues.

Authors:  Laura M Woods; Joseph W Arico; Jeffrey D Frein; Dan L Sackett; Richard E Taylor
Journal:  Int J Mol Sci       Date:  2017-03-17       Impact factor: 5.923

Review 7.  Quest for Efficacious Next-Generation Taxoid Anticancer Agents and Their Tumor-Targeted Delivery.

Authors:  Iwao Ojima; Xin Wang; Yunrong Jing; Changwei Wang
Journal:  J Nat Prod       Date:  2018-02-22       Impact factor: 4.050

8.  Comparison of Epothilone and Taxol Binding in Yeast Tubulin using Molecular Modeling.

Authors:  Vajihe Akbari; Sharareh Moghim; Mohammad Reza Mofid
Journal:  Avicenna J Med Biotechnol       Date:  2011-10
  8 in total

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