Literature DB >> 19841590

Implementation of raltegravir in routine clinical practice: selection criteria for choosing this drug, virologic response rates, and characteristics of failures.

Alexandra U Scherrer1, Viktor von Wyl, Christof A Fux, Milos Opravil, Heiner C Bucher, Aurélie Fayet, Laurent A Decosterd, Bernhard Hirschel, Bettina Khanlari, Sabine Yerly, Thomas Klimkait, Hansjakob Furrer, Bruno Ledergerber, Huldrych F Günthard.   

Abstract

BACKGROUND: Raltegravir (RAL) achieved remarkable virologic suppression rates in randomized-clinical trials, but today efficacy data and factors for treatment failures in a routine clinical care setting are limited.
METHODS: First, factors associated with a switch to RAL were identified with a logistic regression including patients from the Swiss HIV Cohort Study with a history of 3 class failure (n = 423). Second, predictors for virologic outcome were identified in an intent-to-treat analysis including all patients who received RAL. Last observation carried forward imputation was used to determine week 24 response rate (HIV-1 RNA >or= 50 copies/mL).
RESULTS: The predominant factor associated with a switch to RAL in patients with suppressed baseline RNA was a regimen containing enfuvirtide [odds ratio 41.9 (95% confidence interval: 11.6-151.6)]. Efficacy analysis showed an overall response rate of 80.9% (152/188), whereas 71.8% (84/117) and 95.8% (68/71) showed viral suppression when stratified for detectable and undetectable RNA at baseline, respectively. Overall CD4 cell counts increased significantly by 42 cells/microL (P < 0.001). Characteristics of failures were a genotypic sensitivity score of the background regimen <or=1, very low RAL plasma concentrations, poor adherence, and high viral load at baseline.
CONCLUSIONS: Virologic suppression rates in our routine clinical care setting were promising and comparable with data from previously published randomized-controlled trials.

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Year:  2010        PMID: 19841590     DOI: 10.1097/QAI.0b013e3181bca4ec

Source DB:  PubMed          Journal:  J Acquir Immune Defic Syndr        ISSN: 1525-4135            Impact factor:   3.731


  7 in total

1.  Long-term immunologic and virologic responses on raltegravir-containing regimens among ART-experienced participants in the HIV Outpatient Study.

Authors:  Kate Buchacz; Ryan Wiegand; Carl Armon; Joan S Chmiel; Kathleen Wood; John T Brooks; Frank J Palella
Journal:  HIV Clin Trials       Date:  2015-07-01

2.  Effectiveness of integrase strand transfer inhibitors among treatment-experienced patients in a clinical setting.

Authors:  Thibaut Davy-Mendez; Sonia Napravnik; Oksana Zakharova; David A Wohl; Claire E Farel; Joseph J Eron
Journal:  AIDS       Date:  2019-06-01       Impact factor: 4.177

3.  Clinical, virological and immunological responses in Danish HIV patients receiving raltegravir as part of a salvage regimen.

Authors:  Frederik N Engsig; Jan Gerstoft; Gitte Kronborg; Carsten S Larsen; Gitte Pedersen; Anne M Audelin; Louise B Jørgensen; Niels Obel
Journal:  Clin Epidemiol       Date:  2010-08-09       Impact factor: 4.790

4.  Population pharmacokinetic analysis and pharmacogenetics of raltegravir in HIV-positive and healthy individuals.

Authors:  Mona Arab-Alameddine; Aurélie Fayet-Mello; Rubin Lubomirov; Michael Neely; Julia di Iulio; Andrew Owen; Marta Boffito; Matthias Cavassini; Huldrych F Günthard; Katharina Rentsch; Thierry Buclin; Manel Aouri; Amalio Telenti; Laurent Arthur Decosterd; Margalida Rotger; Chantal Csajka
Journal:  Antimicrob Agents Chemother       Date:  2012-02-27       Impact factor: 5.191

5.  Transmitted drug resistance in persons with acute/early HIV-1 in San Francisco, 2002-2009.

Authors:  Vivek Jain; Teri Liegler; Eric Vittinghoff; Wendy Hartogensis; Peter Bacchetti; Lauren Poole; Lisa Loeb; Christopher D Pilcher; Robert M Grant; Steven G Deeks; Frederick M Hecht
Journal:  PLoS One       Date:  2010-12-10       Impact factor: 3.240

Review 6.  Antiretroviral therapy in Indian setting: when & what to start with, when & what to switch to?

Authors:  N Kumarasamy; Atul Patel; Sanjay Pujari
Journal:  Indian J Med Res       Date:  2011-12       Impact factor: 2.375

Review 7.  Next-generation integrase inhibitors : where to after raltegravir?

Authors:  Sharon L Karmon; Martin Markowitz
Journal:  Drugs       Date:  2013-03       Impact factor: 11.431

  7 in total

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