Literature DB >> 1974762

On the fundamental difference in the thermodynamics of agonist and antagonist interactions with beta-adrenergic receptors and the mechanism of entropy-driven binding.

A Miklavc1, D Kocjan, J Mavri, J Koller, D Hadzi.   

Abstract

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Year:  1990        PMID： 1974762     DOI： 10.1016/0006-2952(90)90299-z

Source DB:  PubMed          Journal:  Biochem Pharmacol        ISSN： 0006-2952            Impact factor:   5.858


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  8 in total

1.  Thermodynamically distinct high and low affinity states of the A(1) adenosine receptor induced by G protein coupling and guanine nucleotide ligation states of G proteins.

Authors:  A Lorenzen; L Guerra; F Campi; H Lang; U Schwabe; P A Borea
Journal:  Br J Pharmacol       Date:  2000-06       Impact factor: 8.739

2.  On the stability of nucleic acid structures in solution: enthalpy-entropy compensations, internal rotations and reversibility.

Authors:  M S Searle; D H Williams
Journal:  Nucleic Acids Res       Date:  1993-05-11       Impact factor: 16.971

3.  Thermodynamics and docking of agonists to the β(2)-adrenoceptor determined using [(3)H](R,R')-4-methoxyfenoterol as the marker ligand.

Authors:  Lawrence Toll; Karolina Pajak; Anita Plazinska; Krzysztof Jozwiak; Lucita Jimenez; Joseph A Kozocas; Mary J Tanga; James E Bupp; Irving W Wainer
Journal:  Mol Pharmacol       Date:  2012-03-20       Impact factor: 4.436

4.  The effect of stereochemistry on the thermodynamic characteristics of the binding of fenoterol stereoisomers to the beta(2)-adrenoceptor.

Authors:  Krzysztof Jozwiak; Lawrence Toll; Lucita Jimenez; Anthony Yiu-Ho Woo; Rui-Ping Xiao; Irving W Wainer
Journal:  Biochem Pharmacol       Date:  2010-02-06       Impact factor: 5.858

5.  Toward an estimation of binding constants in aqueous solution: studies of associations of vancomycin group antibiotics.

Authors:  D H Williams; M S Searle; J P Mackay; U Gerhard; R A Maplestone
Journal:  Proc Natl Acad Sci U S A       Date:  1993-02-15       Impact factor: 11.205

6.  [3H]-thioperamide as a radioligand for the histamine H3 receptor in rat cerebral cortex.

Authors:  A Alves-Rodrigues; R Leurs; T S Wu; G D Prell; C Foged; H Timmerman
Journal:  Br J Pharmacol       Date:  1996-08       Impact factor: 8.739

7.  Thermodynamics of antagonist binding to rat muscarinic M2 receptors: antimuscarinics of the pridinol, sila-pridinol, diphenidol and sila-diphenidol type.

Authors:  M Waelbroeck; J Camus; M Tastenoy; G Lambrecht; E Mutschler; M Kropfgans; J Sperlich; F Wiesenberger; R Tacke; J Christophe
Journal:  Br J Pharmacol       Date:  1993-06       Impact factor: 8.739

8.  Thermodynamic analysis of agonist and antagonist binding to the chicken brain melatonin receptor.

Authors:  N W Chong; D Sugden
Journal:  Br J Pharmacol       Date:  1994-01       Impact factor: 8.739
  8 in total

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