Literature DB >> 19646868

Design, synthesis and analgesic properties of novel conformationally-restricted N-acylhydrazones (NAH).

Arthur E Kümmerle1, Marina M Vieira, Martine Schmitt, Ana L P Miranda, Carlos A M Fraga, Jean-Jacques Bourguignon, Eliezer J Barreiro.   

Abstract

A set of six azaheterocycles were designed as conformationally-constrained N-acylhydrazones and tested as analgesics.

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Year:  2009        PMID： 19646868     DOI： 10.1016/j.bmcl.2009.07.075

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  5 in total

Review 1.  Recent advances in the pharmacological diversification of quinazoline/quinazolinone hybrids.

Authors:  Prashant S Auti; Ginson George; Atish T Paul
Journal:  RSC Adv       Date:  2020-11-12       Impact factor: 4.036

Review 2.  MAOS and medicinal chemistry: some important examples from the last years.

Authors:  Nailton M Nascimento-Júnior; Arthur E Kümmerle; Eliezer J Barreiro; Carlos A M Fraga
Journal:  Molecules       Date:  2011-11-07       Impact factor: 4.411

3.  The Discovery of Conformationally Constrained Bicyclic Peptidomimetics as Potent Hepatitis C NS5A Inhibitors.

Authors:  Wieslaw M Kazmierski; Nagaraju Miriyala; David K Johnson; Sam Baskaran
Journal:  ACS Med Chem Lett       Date:  2021-09-15       Impact factor: 4.345

Review 4.  A review exploring biological activities of hydrazones.

Authors:  Garima Verma; Akranth Marella; Mohammad Shaquiquzzaman; Mymoona Akhtar; Mohammad Rahmat Ali; Mohammad Mumtaz Alam
Journal:  J Pharm Bioallied Sci       Date:  2014-04

5.  Biological and quantitative-SAR evaluations, and docking studies of (E)-N -benzylidenebenzohydrazide analogues as potential antibacterial agents.

Authors:  Mohammad Sayed Alam; Sefat Jebin; M Mostafizur Rahman; Md Latiful Bari; Dong-Ung Lee
Journal:  EXCLI J       Date:  2016-06-17       Impact factor: 4.068
  5 in total

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