Literature DB >> 19335274

Targeted therapy in acute myeloid leukaemia: current status and future directions.

Camilla Stapnes1, Bjørn Tore Gjertsen, Håkon Reikvam, Øystein Bruserud.   

Abstract

BACKGROUND: The limit of acceptable toxicity for standard chemotherapeutic drugs used in acute myeloid leukaemia (AML) therapy has been reached. New therapeutic strategies are therefore needed.
OBJECTIVE: This review summarizes development in new strategies, and gives an overview of the clinical status on new drugs for non-promyelocytic AML in adults.
METHODS: Information was principally gathered from the databases ClinicalTrials.gov and PubMed.gov. RESULTS/
CONCLUSION: The major improvements in AML treatment during the last two decades has not been the introduction of new therapeutic agents, but rather the more optimal use of well-known drugs (e.g., high-dose cytarabine therapy, the use of ATRA in maintenance therapy of acute promyelocytic leukaemia) and improvement in the diagnosis and treatment of potentially life-threatening complications in patients treated with allogeneic stem cell transplantation. However, further investigations based on specific targeted therapy and stratification of patients according to knowledge of the individual disease and health status will probably be necessary in future studies of new targeted therapy.

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Year:  2009        PMID: 19335274     DOI: 10.1517/14728220902787628

Source DB:  PubMed          Journal:  Expert Opin Investig Drugs        ISSN: 1354-3784            Impact factor:   6.206


  15 in total

1.  Normal bone marrow signal-transduction profiles: a requisite for enhanced detection of signaling dysregulations in AML.

Authors:  James Marvin; Suchitra Swaminathan; Geoffrey Kraker; Amy Chadburn; James Jacobberger; Charles Goolsby
Journal:  Blood       Date:  2011-01-13       Impact factor: 22.113

2.  Genetic abnormalities and challenges in the treatment of acute myeloid leukemia.

Authors:  C Chandra Kumar
Journal:  Genes Cancer       Date:  2011-02

3.  Dual PI3K/mTOR inhibition shows antileukemic activity in MLL-rearranged acute myeloid leukemia.

Authors:  N Sandhöfer; K H Metzeler; M Rothenberg; T Herold; S Tiedt; V Groiß; M Carlet; G Walter; T Hinrichsen; O Wachter; M Grunert; S Schneider; M Subklewe; A Dufour; S Fröhling; H-G Klein; W Hiddemann; I Jeremias; K Spiekermann
Journal:  Leukemia       Date:  2014-10-17       Impact factor: 11.528

Review 4.  Generating a generation of proteasome inhibitors: from microbial fermentation to total synthesis of salinosporamide a (marizomib) and other salinosporamides.

Authors:  Barbara C Potts; Kin S Lam
Journal:  Mar Drugs       Date:  2010-03-25       Impact factor: 5.118

5.  Marine benthic cyanobacteria contain apoptosis-inducing activity synergizing with daunorubicin to kill leukemia cells, but not cardiomyocytes.

Authors:  Linn Oftedal; Frode Selheim; Matti Wahlsten; Kaarina Sivonen; Stein Ove Døskeland; Lars Herfindal
Journal:  Mar Drugs       Date:  2010-10-14       Impact factor: 5.118

6.  Combined effects of PI3K and SRC kinase inhibitors with imatinib on intracellular calcium levels, autophagy, and apoptosis in CML-PBL cells.

Authors:  Roberto Ciarcia; Sara Damiano; Serena Montagnaro; Ugo Pagnini; Antonio Ruocco; Giuseppe Caparrotti; Danila d'Angelo; Silvia Boffo; Fátima Morales; Flavio Rizzolio; Salvatore Florio; Antonio Giordano
Journal:  Cell Cycle       Date:  2013-08-08       Impact factor: 4.534

Review 7.  Real-time nanoscale proteomic analysis of the novel multi-kinase pathway inhibitor rigosertib to measure the response to treatment of cancer.

Authors:  Alice C Fan; Jennifer J O'Rourke; Dave R Praharaj; Dean W Felsher
Journal:  Expert Opin Investig Drugs       Date:  2013-08-12       Impact factor: 6.206

8.  The novel tyrosine kinase inhibitor AKN-028 has significant antileukemic activity in cell lines and primary cultures of acute myeloid leukemia.

Authors:  A Eriksson; M Hermanson; M Wickström; E Lindhagen; C Ekholm; A Jenmalm Jensen; A Löthgren; F Lehmann; R Larsson; V Parrow; M Höglund
Journal:  Blood Cancer J       Date:  2012-08-03       Impact factor: 11.037

9.  Inhibition of Mammalian target of rapamycin in human acute myeloid leukemia cells has diverse effects that depend on the environmental in vitro stress.

Authors:  Anita Ryningen; Håkon Reikvam; Ina Nepstad; Kristin Paulsen Rye; Oystein Bruserud
Journal:  Bone Marrow Res       Date:  2012-10-02

10.  Pharmacological targeting of the PI3K/mTOR pathway alters the release of angioregulatory mediators both from primary human acute myeloid leukemia cells and their neighboring stromal cells.

Authors:  Håkon Reikvam; Ina Nepstad; Øystein Bruserud; Kimberley Joanne Hatfield
Journal:  Oncotarget       Date:  2013-06
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