Literature DB >> 1928875

Simulated acetaminophen overdose: pharmacokinetics and effectiveness of activated charcoal.

S R Rose1, R L Gorman, G M Oderda, W Klein-Schwartz, W A Watson.   

Abstract

STUDY
OBJECTIVE: To determine the absorption rate of a supratherapeutic dose of acetaminophen elixir and compare the effect of activated charcoal (AC) given at different time intervals on preventing acetaminophen absorption.
DESIGN: Randomized, nonblinded, crossover controlled study.
SETTING: A certified regional poison control center. PARTICIPANTS: Ten healthy, adult male volunteers from 21 to 39 years old.
INTERVENTIONS: Each subject received 5 g acetaminophen (elixir) on four occasions: a control phase plus 30 g of AC administered 15, 30, or 120 minutes after acetaminophen. Serum acetaminophen levels were obtained during the control phase only, and 24-hour urine collections were obtained during all four phases.
MEASUREMENTS AND MAIN RESULTS: The highest serum acetaminophen levels were measured 1.4 +/- 0.52 hours after ingestion, and absorption was 97% complete by a mean of 2.05 hours. The administration of AC at 15, 30, and 120 minutes after acetaminophen reduced urinary recovery of acetaminophen and metabolites by 48%, 44%, and 33%, respectively.
CONCLUSION: AC significantly reduces urinary recovery but not absorption of acetaminophen when administered two hours after acetaminophen elixir.

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Year:  1991        PMID: 1928875     DOI: 10.1016/s0196-0644(05)81353-8

Source DB:  PubMed          Journal:  Ann Emerg Med        ISSN: 0196-0644            Impact factor:   5.721


  3 in total

1.  Effectiveness of delayed activated charcoal administration in simulated paracetamol (acetaminophen) overdose.

Authors:  P J Yeates; S H Thomas
Journal:  Br J Clin Pharmacol       Date:  2000-01       Impact factor: 4.335

2.  Gastrointestinal decontamination in the acutely poisoned patient.

Authors:  Timothy E Albertson; Kelly P Owen; Mark E Sutter; Andrew L Chan
Journal:  Int J Emerg Med       Date:  2011-10-12

Review 3.  Gastric decontaminating procedures: is it time to call a stop?

Authors:  J P Saetta
Journal:  J R Soc Med       Date:  1993-07       Impact factor: 18.000

  3 in total

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