Literature DB >> 19092711

Raloxifene use in clinical practice: efficacy and safety.

Steven R Goldstein1, Claire S Duvernoy, Joaquim Calaf, Jonathan D Adachi, John L Mershon, Sherie A Dowsett, Donato Agnusdei, Cynthia A Stuenkel.   

Abstract

OBJECTIVE AND METHODS: In this article, we provide an interdisciplinary concise review of the effects of raloxifene on breast, bone, and reproductive organs, as well as the adverse events that may be associated with its use.
RESULTS: Raloxifene has been shown to prevent osteoporosis in postmenopausal women (PMW) with low bone mass and prevent vertebral fractures in those with osteoporosis/low bone mass; it has not been shown to reduce the risk of nonvertebral fractures. Raloxifene reduces the risk of invasive breast cancer in PMW with osteoporosis or at high risk of breast cancer. The risk of venous thromboembolism has been consistently shown to be increased with raloxifene, so it should not be used in women at high risk of venous thromboembolism. Although raloxifene does not increase, nor decrease, the risk of coronary or stroke events overall, in the raloxifene trial of PMW at increased risk of coronary events, the incidence of fatal stroke was higher in women assigned raloxifene versus placebo.
CONCLUSIONS: Based on its approved indications, it is appropriate to prescribe raloxifene to prevent or treat osteoporosis, as well as to reduce the risk of invasive breast cancer in PMW with osteoporosis or at high risk of breast cancer. Women at increased risk of both fracture and invasive breast cancer are those most likely to receive a dual benefit with raloxifene. Decision making must involve the incorporation of the woman's personal feelings about the risks and benefits of raloxifene therapy, balanced with her interest in reducing risk of fractures and breast cancer through pharmacological intervention.

Entities:  

Mesh:

Substances:

Year:  2009        PMID: 19092711     DOI: 10.1097/gme.0b013e3181883dae

Source DB:  PubMed          Journal:  Menopause        ISSN: 1072-3714            Impact factor:   2.953


  14 in total

Review 1.  Recommendations for raloxifene use in daily clinical practice in the Swiss setting.

Authors:  Kurt Lippuner; P A Buchard; C De Geyter; B Imthurn; O Lamy; M Litschgi; F Luzuy; K Schiessl; P Stute; M Birkhäuser
Journal:  Eur Spine J       Date:  2012-06-28       Impact factor: 3.134

Review 2.  Strontium ranelate: a review of its use in the treatment of postmenopausal osteoporosis.

Authors:  Emma D Deeks; Sohita Dhillon
Journal:  Drugs       Date:  2010-04-16       Impact factor: 9.546

3.  Safety and effectiveness profile of raloxifene in long-term, prospective, postmarketing surveillance.

Authors:  Noriko Iikuni; Etsuro Hamaya; Shigeru Nihojima; Shunji Yokoyama; Wakana Goto; Masanori Taketsuna; Akimitsu Miyauchi; Hideaki Sowa
Journal:  J Bone Miner Metab       Date:  2012-07-03       Impact factor: 2.626

Review 4.  Advances in Our Understanding of the Mechanism of Action of Drugs (including Traditional Chinese Medicines) for the Intervention and Treatment of Osteoporosis.

Authors:  Junjie Lu; Desheng Hu; Chen Ma; Bo Shuai
Journal:  Front Pharmacol       Date:  2022-06-14       Impact factor: 5.988

Review 5.  Signaling, physiological functions and clinical relevance of the G protein-coupled estrogen receptor GPER.

Authors:  Eric R Prossnitz; Matthias Barton
Journal:  Prostaglandins Other Lipid Mediat       Date:  2009-05-13       Impact factor: 3.072

6.  The short-term effects of estradiol, raloxifene, and a phytoestrogen in women with perimenopausal depression.

Authors:  Peter J Schmidt; Shau-Ming Wei; Pedro E Martinez; Rivka R Ben Dor; Gioia M Guerrieri; Paula P Palladino; Veronica L Harsh; Howard J Li; Paul Wakim; Lynnette K Nieman; David R Rubinow
Journal:  Menopause       Date:  2021-01-15       Impact factor: 3.310

Review 7.  Emerging therapies for the treatment of osteoporosis.

Authors:  Garima Bhutani; Mahesh Chander Gupta
Journal:  J Midlife Health       Date:  2013-07

Review 8.  The Tissue-Selective Estrogen Complex: A Review of Current Evidence.

Authors:  Rinu Pazhekattu; Arthur N Lau; Jonathan D Adachi
Journal:  Rheumatol Ther       Date:  2015-05-20

9.  Combined oral administration of bovine collagen peptides with calcium citrate inhibits bone loss in ovariectomized rats.

Authors:  JunLi Liu; YiHu Wang; ShuJun Song; XiJie Wang; YaYa Qin; ShaoYan Si; YanChuan Guo
Journal:  PLoS One       Date:  2015-08-10       Impact factor: 3.240

10.  Cardiovascular risk factor analysis in patients with a recent clinical fracture at the fracture liaison service.

Authors:  Caroline E Wyers; Lisanne Vranken; Robert Y van der Velde; Piet P M M Geusens; Heinrich M J Janzing; J Wim Morrenhof; Joop P W van den Bergh
Journal:  Biomed Res Int       Date:  2014-08-27       Impact factor: 3.411

View more

北京卡尤迪生物科技股份有限公司 © 2022-2023.