Literature DB >> 19065645

Assessing the bioisosterism of the trifluoromethyl group with a protease probe.

Monika Jagodzinska1, Florent Huguenot, Gabriele Candiani, Matteo Zanda.   

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Year:  2009        PMID： 19065645     DOI： 10.1002/cmdc.200800321

Source DB:  PubMed          Journal:  ChemMedChem        ISSN： 1860-7179            Impact factor:   3.466


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  10 in total

1.  Palladium-catalyzed coupling reactions on functionalized 2-trifluoromethyl-4-chromenone scaffolds. Synthesis of highly functionalized trifluoromethyl-heterocycles.

Authors:  Javier Izquierdo; Atul D Jain; Sarki A Abdulkadir; Gary E Schiltz
Journal:  Synthesis (Stuttg)       Date:  2019-03       Impact factor: 3.157

2.  Carba Analogues of Flupirtine and Retigabine with Improved Oxidation Resistance and Reduced Risk of Quinoid Metabolite Formation.

Authors:  Konrad W Wurm; Frieda-Marie Bartz; Lukas Schulig; Anja Bodtke; Patrick J Bednarski; Andreas Link
Journal:  ChemMedChem       Date:  2022-07-07       Impact factor: 3.540

3.  Electronically Activated Organoboron Catalysts for Enantioselective Propargyl Addition to Trifluoromethyl Ketones.

Authors:  Nicholas W Mszar; Malte S Mikus; Sebastian Torker; Fredrik Haeffner; Amir H Hoveyda
Journal:  Angew Chem Int Ed Engl       Date:  2017-06-21       Impact factor: 15.336

4.  19F-Tagged metal binding pharmacophores for NMR screening of metalloenzymes.

Authors:  Kathleen E Prosser; Alysia J Kohlbrand; Hyeonglim Seo; Mark Kalaj; Seth M Cohen
Journal:  Chem Commun (Camb)       Date:  2021-05-18       Impact factor: 6.222

5.  Study on a Three-Step Rapid Assembly of Zolpidem and Its Fluorinated Analogues Employing Microwave-Assisted Chemistry.

Authors:  Nikola Fajkis; Monika Marcinkowska; Beata Gryzło; Anna Krupa; Marcin Kolaczkowski
Journal:  Molecules       Date:  2020-07-10       Impact factor: 4.411

6.  New methodology for the synthesis of thiobarbiturates mediated by manganese(III) acetate.

Authors:  Ahlem Bouhlel; Christophe Curti; Patrice Vanelle
Journal:  Molecules       Date:  2012-04-10       Impact factor: 4.411

7.  Crystal structures and antifungal activities of fluorine-containing thioureido complexes with nickel(II).

Authors:  Chun Li; Wen Yang; Huanhuan Liu; Mengying Li; Weiqun Zhou; Juan Xie
Journal:  Molecules       Date:  2013-12-17       Impact factor: 4.411

8.  Catalytic enantioselective addition of organoboron reagents to fluoroketones controlled by electrostatic interactions.

Authors:  KyungA Lee; Daniel L Silverio; Sebastian Torker; Daniel W Robbins; Fredrik Haeffner; Farid W van der Mei; Amir H Hoveyda
Journal:  Nat Chem       Date:  2016-05-23       Impact factor: 24.427

9.  Preparative Method for Asymmetric Synthesis of (S)-2-Amino-4,4,4-trifluorobutanoic Acid.

Authors:  Jianlin Han; Ryosuke Takeda; Xinyi Liu; Hiroyuki Konno; Hidenori Abe; Takahiro Hiramatsu; Hiroki Moriwaki; Vadim A Soloshonok
Journal:  Molecules       Date:  2019-12-10       Impact factor: 4.411

10.  Design and synthesis of pyrazolopyridine derivatives as sphingosine 1-phosphate receptor 2 ligands.

Authors:  Zonghua Luo; Xuyi Yue; Hao Yang; Hui Liu; Robyn S Klein; Zhude Tu
Journal:  Bioorg Med Chem Lett       Date:  2017-12-06       Impact factor: 2.823
  10 in total

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