Literature DB >> 19041149

The profile of mutational clusters associated with lamivudine resistance can be constrained by HBV genotypes.

Valentina Svicher1, Caterina Gori, Maria Trignetti, Michela Visca, Valeria Micheli, Martina Bernassola, Romina Salpini, Guido Gubertini, Roberta Longo, Fosca Niero, Francesca Ceccherini-Silberstein, Giuseppe Maria De Sanctis, Alberto Spanò, Giuseppina Cappiello, Carlo Federico Perno.   

Abstract

BACKGROUND/AIMS: To investigate the different clusters of mutations associated with lamivudine resistance in HBV genotypes D and A.
METHODS: HBV reverse transcriptase sequences of 89 HBV-infected patients failing lamivudine treatment were analyzed. The association of mutations with HBV genotypes was assessed by Chi-Squared test and multivariate logistic regression analysis. Covariate analysis was based on hierarchical clustering.
RESULTS: In genotype A, the rtM204V (prevalence: 68.2%) was the main sign of lamivudine failure. Multivariate analysis confirmed that genotype A is the only predictor for rtM204V emergence (OR: 14.5 [95% CI: 1.3-158], P=0.02). Covariate analysis showed that rtM204V clusters with rtL180M, rtL229V (corresponding to sF220L in the HBsAg), and, interestingly, with HBsAg mutation sS207N (bootstrap=0.95). Both sF220L and sS207N co-localized in the fourth transmembrane HBsAg domain. In contrast, in genotype D the primary mutations rtM204V and rtM204I occurred with similar prevalence (39.1% versus 45.3%, P=0.47), and showed a distinct pattern of compensatory mutations. rtM204V clusters with mutations localized in the RT-B domain (rtV173L, rtL180M, and rtT184A/S) (bootstrap=0.94), while rtM204I clusters with mutations localized in the RT-A domain (rtS53N, rtT54Y, and rtL80I/V) (bootstrap=0.96) (without associations with HBsAg specific mutations).
CONCLUSIONS: HBV genotype plays an important role in driving RT evolution under lamivudine treatment, and thus can be relevant for therapeutic sequencing, immunological response and disease progression.

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Year:  2008        PMID: 19041149     DOI: 10.1016/j.jhep.2008.07.038

Source DB:  PubMed          Journal:  J Hepatol        ISSN: 0168-8278            Impact factor:   25.083


  9 in total

1.  High rates of chronic HBV genotype E infection in a group of migrants in Italy from West Africa: Virological characteristics associated with poor immune clearance.

Authors:  Vincenzo Malagnino; Romina Salpini; Gaetano Maffongelli; Arianna Battisti; Lavinia Fabeni; Lorenzo Piermatteo; Luna Colagrossi; Vanessa Fini; Alessandra Ricciardi; Cesare Sarrecchia; Carlo Federico Perno; Massimo Andreoni; Valentina Svicher; Loredana Sarmati
Journal:  PLoS One       Date:  2018-03-29       Impact factor: 3.240

2.  Immune-escape mutations and stop-codons in HBsAg develop in a large proportion of patients with chronic HBV infection exposed to anti-HBV drugs in Europe.

Authors:  Luna Colagrossi; Lucas E Hermans; Romina Salpini; Domenico Di Carlo; Suzan D Pas; Marta Alvarez; Ziv Ben-Ari; Greet Boland; Bianca Bruzzone; Nicola Coppola; Carole Seguin-Devaux; Tomasz Dyda; Federico Garcia; Rolf Kaiser; Sukran Köse; Henrik Krarup; Ivana Lazarevic; Maja M Lunar; Sarah Maylin; Valeria Micheli; Orna Mor; Simona Paraschiv; Dimitros Paraskevis; Mario Poljak; Elisabeth Puchhammer-Stöckl; François Simon; Maja Stanojevic; Kathrine Stene-Johansen; Nijaz Tihic; Pascale Trimoulet; Jens Verheyen; Adriana Vince; Snjezana Zidovec Lepej; Nina Weis; Tülay Yalcinkaya; Charles A B Boucher; Annemarie M J Wensing; Carlo F Perno; Valentina Svicher
Journal:  BMC Infect Dis       Date:  2018-06-01       Impact factor: 3.090

3.  Key mutations in the C-terminus of the HBV surface glycoprotein correlate with lower HBsAg levels in vivo, hinder HBsAg secretion in vitro and reduce HBsAg structural stability in the setting of HBeAg-negative chronic HBV genotype-D infection.

Authors:  Romina Salpini; Arianna Battisti; Lorenzo Piermatteo; Luca Carioti; Olympia E Anastasiou; Upkar S Gill; Domenico Di Carlo; Luna Colagrossi; Leonardo Duca; Ada Bertoli; Katia Yu La Rosa; Lavinia Fabeni; Alessandra Iuvara; Vincenzo Malagnino; Carlotta Cerva; Miriam Lichtner; Claudio M Mastroianni; Giuseppe Maria De Sanctis; Maurizio Paoloni; Massimo Marignani; Caterina Pasquazzi; Nerio Iapadre; Giustino Parruti; Jacopo Vecchiet; Loredana Sarmati; Massimo Andreoni; Mario Angelico; Sandro Grelli; Patrick T Kennedy; Jens Verheyen; Stefano Aquaro; Francesca Ceccherini Silberstein; Carlo Federico Perno; Valentina Svicher
Journal:  Emerg Microbes Infect       Date:  2020-12       Impact factor: 7.163

4.  Key genetic elements, single and in clusters, underlying geographically dependent SARS-CoV-2 genetic adaptation and their impact on binding affinity for drugs and immune control.

Authors:  Romina Salpini; Mohammad Alkhatib; Giosuè Costa; Lorenzo Piermatteo; Francesca Alessandra Ambrosio; Velia Chiara Di Maio; Rossana Scutari; Leonardo Duca; Giulia Berno; Lavinia Fabeni; Stefano Alcaro; Francesca Ceccherini-Silberstein; Anna Artese; Valentina Svicher
Journal:  J Antimicrob Chemother       Date:  2021-01-19       Impact factor: 5.790

5.  Characterization of antiviral resistance mutations among the Eastern Indian Hepatitis B virus infected population.

Authors:  Rajesh Panigrahi; Avik Biswas; Binay Krishna De; Sekhar Chakrabarti; Runu Chakravarty
Journal:  Virol J       Date:  2013-02-14       Impact factor: 4.099

6.  Mutational analysis of reverse transcriptase and surface proteins of patients with partial virological response during mono and combination antiviral therapies in genotype D chronic hepatitis B.

Authors:  Mostafa Mahabadi; Seyed Moayed Alavian; Mehdi Norouzi; Hossein Keyvani; Mahmood Mahmoudi; Seyed Mohammad Jazayeri
Journal:  Electron Physician       Date:  2016-06-25

7.  Prevalence of Single and Multiple Natural NS3, NS5A and NS5B Resistance-Associated Substitutions in Hepatitis C Virus Genotypes 1-4 in Italy.

Authors:  Ada Bertoli; Maria Chiara Sorbo; Marianna Aragri; Ilaria Lenci; Elisabetta Teti; Ennio Polilli; Velia Chiara Di Maio; Laura Gianserra; Elisa Biliotti; Chiara Masetti; Carlo F Magni; Sergio Babudieri; Laura A Nicolini; Martina Milana; Pierluigi Cacciatore; Loredana Sarmati; Adriano Pellicelli; Stefania Paolucci; Antonio Craxì; Filomena Morisco; Valeria Pace Palitti; Massimo Siciliano; Nicola Coppola; Nerio Iapadre; Massimo Puoti; Giuliano Rizzardini; Gloria Taliani; Caterina Pasquazzi; Massimo Andreoni; Giustino Parruti; Mario Angelico; Carlo Federico Perno; Valeria Cento; Francesca Ceccherini-Silberstein
Journal:  Sci Rep       Date:  2018-06-12       Impact factor: 4.379

Review 8.  Naturally occurring hepatitis B virus reverse transcriptase mutations related to potential antiviral drug resistance and liver disease progression.

Authors:  Yu-Min Choi; So-Young Lee; Bum-Joon Kim
Journal:  World J Gastroenterol       Date:  2018-04-28       Impact factor: 5.742

9.  Mutational characterization of HBV reverse transcriptase gene and the genotype-phenotype correlation of antiviral resistance among Chinese chronic hepatitis B patients.

Authors:  Ya Fu; Songhang Wu; Yuhai Hu; Tianbin Chen; Yongbin Zeng; Can Liu; Qishui Ou
Journal:  Emerg Microbes Infect       Date:  2020-12       Impact factor: 7.163

  9 in total

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