Literature DB >> 18973169

Bisphosphonated benzoxazinorifamycin prodrugs for the prevention and treatment of osteomyelitis.

Ranga Reddy1, Evelyne Dietrich, Yanick Lafontaine, Tom J Houghton, Odette Belanger, Anik Dubois, Francis F Arhin, Ingrid Sarmiento, Ibtihal Fadhil, Karine Laquerre, Valerie Ostiguy, Dario Lehoux, Gregory Moeck, Thomas R Parr, Adel Rafai Far.   

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Year:  2008        PMID: 18973169     DOI: 10.1002/cmdc.200800255

Source DB:  PubMed          Journal:  ChemMedChem        ISSN: 1860-7179            Impact factor:   3.466


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  7 in total

1.  1-(Fluoroalkylidene)-1,1-bisphosphonic acids are potent and selective inhibitors of the enzymatic activity of Toxoplasma gondii farnesyl pyrophosphate synthase.

Authors:  Sergio H Szajnman; Valeria S Rosso; Leena Malayil; Alyssa Smith; Silvia N J Moreno; Roberto Docampo; Juan B Rodriguez
Journal:  Org Biomol Chem       Date:  2012-01-03       Impact factor: 3.876

2.  In Vitro and In Vivo Activities of Sulfur-Containing Linear Bisphosphonates against Apicomplexan Parasites.

Authors:  Sergio H Szajnman; Tamila Galaka; Zhu-Hong Li; Catherine Li; Nathan M Howell; María N Chao; Boris Striepen; Vasant Muralidharan; Silvia N J Moreno; Juan B Rodriguez
Journal:  Antimicrob Agents Chemother       Date:  2017-01-24       Impact factor: 5.191

3.  Design, synthesis, calorimetry, and crystallographic analysis of 2-alkylaminoethyl-1,1-bisphosphonates as inhibitors of Trypanosoma cruzi farnesyl diphosphate synthase.

Authors:  Srinivas Aripirala; Sergio H Szajnman; Jean Jakoncic; Juan B Rodriguez; Roberto Docampo; Sandra B Gabelli; L Mario Amzel
Journal:  J Med Chem       Date:  2012-07-05       Impact factor: 7.446

4.  Synergistic Activity between Statins and Bisphosphonates against Acute Experimental Toxoplasmosis.

Authors:  Zhu-Hong Li; Catherine Li; Sergio H Szajnman; Juan B Rodriguez; Silvia N J Moreno
Journal:  Antimicrob Agents Chemother       Date:  2017-07-25       Impact factor: 5.191

5.  Design, synthesis and biological evaluation of sulfur-containing 1,1-bisphosphonic acids as antiparasitic agents.

Authors:  Marion Recher; Alejandro P Barboza; Zhu-Hong Li; Melina Galizzi; Mariana Ferrer-Casal; Sergio H Szajnman; Roberto Docampo; Silvia N J Moreno; Juan B Rodriguez
Journal:  Eur J Med Chem       Date:  2012-12-20       Impact factor: 6.514

6.  Antiparasitic Activity of Sulfur- and Fluorine-Containing Bisphosphonates against Trypanosomatids and Apicomplexan Parasites.

Authors:  Tamila Galaka; Mariana Ferrer Casal; Melissa Storey; Catherine Li; María N Chao; Sergio H Szajnman; Roberto Docampo; Silvia N J Moreno; Juan B Rodriguez
Journal:  Molecules       Date:  2017-01-04       Impact factor: 4.411

Review 7.  Bisphosphonate conjugation for bone specific drug targeting.

Authors:  Kristen B Farrell; Alexander Karpeisky; Douglas H Thamm; Shawn Zinnen
Journal:  Bone Rep       Date:  2018-07-03
  7 in total

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