Literature DB >> 18959421

Synthesis and biological activities of novel pyrazole oxime derivatives containing a 2-chloro-5-thiazolyl moiety.

Hong Dai1, Yong-Qiang Li, Ding Du, Xue Qin, Xin Zhang, Hai-Bo Yu, Jian-Xin Fang.   

Abstract

A series of novel pyrazole oxime derivatives containing a 2-chloro-5-thiazolyl moiety were synthesized. Their structures were confirmed by (1)H NMR, (13)C NMR, and elemental analysis. The preliminary bioassays showed that all of the title compounds had low acaricidal activity against Tetranychus cinnabarinus . However, most of them exhibited excellent insecticidal activity against Aphis medicagini at the dosage of 0.5 mg/mL, and some compounds still showed good insecticidal activity against A. medicagini even at the dosage of 0.2 mg/mL. Meanwhile, some title compounds displayed fungicidal and plant growth regulatory activities.

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Year:  2008        PMID: 18959421     DOI: 10.1021/jf802429x

Source DB:  PubMed          Journal:  J Agric Food Chem        ISSN: 0021-8561            Impact factor:   5.279


  6 in total

1.  Pyrazolylthiazole as DeltaF508-cystic fibrosis transmembrane conductance regulator correctors with improved hydrophilicity compared to bithiazoles.

Authors:  Long Ye; John M Knapp; Panjamaporn Sangwung; James C Fettinger; A S Verkman; Mark J Kurth
Journal:  J Med Chem       Date:  2010-05-13       Impact factor: 7.446

2.  Thermal electron-transfer-induced oxidation of 2-pyrazolines.

Authors:  Hamid Reza Memarian; Reza Minakar
Journal:  Mol Divers       Date:  2019-02-02       Impact factor: 2.943

3.  Synthesis and Bioactivities of Novel Pyrazole Oxime Derivatives Containing a 5-Trifluoromethylpyridyl Moiety.

Authors:  Hong Dai; Jia Chen; Hong Li; Baojiang Dai; Haibing He; Yuan Fang; Yujun Shi
Journal:  Molecules       Date:  2016-02-27       Impact factor: 4.411

4.  Novel Pyridyl-Oxazole Carboxamides: Toxicity Assay Determination in Fungi and Zebrafish Embryos.

Authors:  Shu Chen; Dong-Lin Zhang; Chao-Li Ren; Wen-Qian Zou; Xiao-Yu Tian; Xiao-Hua Du; Cheng-Xia Tan
Journal:  Molecules       Date:  2021-06-25       Impact factor: 4.411

5.  Evaluation of etoxazole against insects and acari in vegetables in China.

Authors:  Yongqiang Li; Na Yang; Xingcun Wei; Yun Ling; Xinling Yang; Qingmin Wang
Journal:  J Insect Sci       Date:  2014       Impact factor: 1.857

6.  Uses of cyanoacetylhydrazine in heterocyclic synthesis: novel synthesis of pyrazole derivatives with anti-tumor activities.

Authors:  Rafat M Mohareb; Nahed N E El-Sayed; Mahmoud A Abdelaziz
Journal:  Molecules       Date:  2012-07-12       Impact factor: 4.411

  6 in total

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