Literature DB >> 1895308

Potent, orally active imidazo[4,5-b]pyridine-based angiotensin II receptor antagonists.

N B Mantlo1, P K Chakravarty, D L Ondeyka, P K Siegl, R S Chang, V J Lotti, K A Faust, T B Chen, T W Schorn, C S Sweet.   

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Year:  1991        PMID： 1895308     DOI： 10.1021/jm00113a035

Source DB:  PubMed          Journal:  J Med Chem        ISSN： 0022-2623            Impact factor:   7.446


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  6 in total

1.  Derivation of a 3D pharmacophore model for the angiotensin-II site one receptor.

Authors:  K Prendergast; K Adams; W J Greenlee; R B Nachbar; A A Patchett; D J Underwood
Journal:  J Comput Aided Mol Des       Date:  1994-10       Impact factor: 3.686

2.  A 3D QSAR approach to the search for geometrical similarity in a series of nonpeptide angiotensin II receptor antagonists.

Authors:  L Belvisi; G Bravi; C Scolastico; A Vulpetti; A Salimbeni; R Todeschini
Journal:  J Comput Aided Mol Des       Date:  1994-04       Impact factor: 3.686

3.  Characterization of the angiotensin II AT1 receptor subtype involved in DNA synthesis in cultured vascular smooth muscle cells.

Authors:  V Briand; L Riva; A M Galzin
Journal:  Br J Pharmacol       Date:  1994-08       Impact factor: 8.739

4.  Pharmacological profile of valsartan: a potent, orally active, nonpeptide antagonist of the angiotensin II AT1-receptor subtype.

Authors:  L Criscione; M de Gasparo; P Bühlmayer; S Whitebread; H P Ramjoué; J Wood
Journal:  Br J Pharmacol       Date:  1993-10       Impact factor: 8.739

Review 5.  Rational Design and Synthesis of AT1R Antagonists.

Authors:  Nikitas Georgiou; Vasileios K Gkalpinos; Spyridon D Katsakos; Stamatia Vassiliou; Andreas G Tzakos; Thomas Mavromoustakos
Journal:  Molecules       Date:  2021-05-14       Impact factor: 4.411

6.  Tautomerization, molecular structure, transition state structure, and vibrational spectra of 2-aminopyridines: a combined computational and experimental study.

Authors:  Jamelah S Al-Otaibi
Journal:  Springerplus       Date:  2015-10-09
  6 in total

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