Literature DB >> 18945255

Clinical trial: pilot study of metformin for the treatment of non-alcoholic steatohepatitis.

R Loomba1, G Lutchman, D E Kleiner, M Ricks, J J Feld, B B Borg, A Modi, P Nagabhyru, A E Sumner, T J Liang, J H Hoofnagle.   

Abstract

BACKGROUND: Non-alcoholic steatohepatitis (NASH) is a form of progressive fatty liver disease that is strongly associated with insulin resistance, which suggests that insulin sensitizing agents such as metformin may be beneficial for NASH. AIM: To assess the effects of metformin on insulin sensitivity, body composition, serum alanine aminotransferase (ALT) levels and liver histology in patients with NASH.
METHODS: Patients underwent liver biopsy, metabolic profiling and imaging studies before and at the end 48 weeks of metformin (2000 mg/day) therapy. The primary endpoint was a three-point improvement in the histological NASH activity index.
RESULTS: Of 28 patients enrolled, 26 (13 females; average age 44 years) completed 48 weeks of treatment and underwent repeat metabolic studies, imaging and liver biopsy. Thirty per cent achieved a histological response. Most patients lost weight, the average being 6 kg. There was a marked association between weight loss and improvements in NASH activity index and ALT levels (both, P < 0.01). Insulin sensitivity also improved, but the degree of change did not correlate with histological improvement.
CONCLUSION: Metformin leads to improvements in liver histology and ALT levels in 30% of patients with NASH, probably by its effects in causing weight loss.

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Year:  2008        PMID: 18945255      PMCID: PMC2990687          DOI: 10.1111/j.1365-2036.2008.03869.x

Source DB:  PubMed          Journal:  Aliment Pharmacol Ther        ISSN: 0269-2813            Impact factor:   8.171


  25 in total

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2.  Beneficial effects of metformin in normoglycemic morbidly obese adolescents.

Authors:  J P Kay; R Alemzadeh; G Langley; L D'Angelo; P Smith; S Holshouser
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