Literature DB >> 18842403

Synthesis and antibacterial activities of novel oxazolidinones having cyclic sulfonamide moieties.

Seong Jong Kim1, Seoung Jong Kim, Myung-Ho Jung, Kyung Ho Yoo, Jung-Hyuck Cho, Chang-Hyun Oh.   

Abstract

The synthesis of a new series of oxazolidinones having cyclic sulfonamide moieties is described. Their in vitro antibacterial activities against both Gram-positive and Gram-negative bacteria were tested and the effect of substituents on the oxazolidinone ring was investigated. A particular compound 15g having [1,2,5]thiadiazolidin-1,1-dioxide moiety showed the most potent antibacterial activity.

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Year:  2008        PMID： 18842403     DOI： 10.1016/j.bmcl.2008.09.034

Source DB:  PubMed          Journal:  Bioorg Med Chem Lett        ISSN： 0960-894X            Impact factor:   2.823


  8 in total

1.  Complementary regioselectivity in the Cu(I)-catalyzed diamination of conjugated dienes to form cyclic sulfamides.

Authors:  Richard G Cornwall; Baoguo Zhao; Yian Shi
Journal:  Org Lett       Date:  2010-12-30       Impact factor: 6.005

2.  Asymmetric Palladium-Catalyzed Alkene Carboamination Reactions for the Synthesis of Cyclic Sulfamides.

Authors:  Zachary J Garlets; Kaia R Parenti; John P Wolfe
Journal:  Chemistry       Date:  2016-03-10       Impact factor: 5.236

3.  Synthesis and Selective Functionalization of Thiadiazine 1,1-Dioxides with Efficacy in a Model of Huntington's Disease.

Authors:  Leila Terrab; Christopher J Rosenker; Lisa Johnstone; Linh K Ngo; Li Zhang; Nathaniel F Ware; Bettina Miller; Andrea Z Topacio; Sara Sannino; Jeffrey L Brodsky; Peter Wipf
Journal:  ACS Med Chem Lett       Date:  2020-02-20       Impact factor: 4.345

4.  Photochemically-Mediated, Nickel-Catalyzed Synthesis of N-(Hetero)aryl Sulfamate Esters.

Authors:  J Miles Blackburn; Anastasia L Gant Kanegusuku; Georgia E Scott; Jennifer L Roizen
Journal:  Org Lett       Date:  2019-08-22       Impact factor: 6.005

5.  Influence of catalyst structure and reaction conditions on anti- versus syn-aminopalladation pathways in Pd-catalyzed alkene carboamination reactions of N-allylsulfamides.

Authors:  Ryan M Fornwald; Jonathan A Fritz; John P Wolfe
Journal:  Chemistry       Date:  2014-06-17       Impact factor: 5.236

6.  Catalytic asymmetric synthesis of cyclic sulfamides from conjugated dienes.

Authors:  Richard G Cornwall; Baoguo Zhao; Yian Shi
Journal:  Org Lett       Date:  2013-01-30       Impact factor: 6.005

7.  Synthesis, in silico study (DFT, ADMET) and crystal structure of novel sulfamoyloxy-oxazolidinones: Interaction with SARS-CoV-2.

Authors:  Abdeslem Bouzina; Malika Berredjem; Sofiane Bouacida; Khaldoun Bachari; Christelle Marminon; Marc Le Borgne; Zouhair Bouaziz; Yousra Ouafa Bouone
Journal:  J Mol Struct       Date:  2022-02-05       Impact factor: 3.841

8.  Efficient Routes to a Diverse Array of Amino Alcohol-Derived Chiral Fragments.

Authors:  Sina Haftchenary; Shawn D Nelson; Laura Furst; Sivaraman Dandapani; Steven J Ferrara; Žarko V Bošković; Samuel Figueroa Lazú; Adrian M Guerrero; Juan C Serrano; DeMarcus K Crews; Cristina Brackeen; Jeffrey Mowat; Thomas Brumby; Marcus Bauser; Stuart L Schreiber; Andrew J Phillips
Journal:  ACS Comb Sci       Date:  2016-08-12       Impact factor: 3.784
  8 in total

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