Literature DB >> 18756533

Clofarabine combinations as acute myeloid leukemia salvage therapy.

Stefan Faderl1, Alessandra Ferrajoli, William Wierda, Xuelin Huang, Srdan Verstovsek, Farhad Ravandi, Zeev Estrov, Gautam Borthakur, Monica Kwari, Hagop M Kantarjian.   

Abstract

BACKGROUND: Outcome of patients with relapsed acute myeloid leukemia (AML) remains unsatisfactory. Clofarabine is a nucleoside analog with activity in adult AML. Combinations with cytarabine in AML are feasible and effective. Idarubicin is another active AML drug, which has not yet been tested with clofarabine.
METHODS: The authors therefore designed a phase I study of clofarabine +/- cytarabine, plus idarubicin. Patients with primary refractory or first-relapse AML were assigned to either clofarabine plus idarubicin (CI) if previously exposed to cytarabine with a response lasting <12 months, or clofarabine and idarubicin plus cytarabine (CIA) for responses > or = 12 months, or if never exposed to cytarabine. A standard "3 + 3" phase 1 design was followed to define maximum tolerated dose (MTD). Forty-four patients were treated (23 CI; 21 CIA).
RESULTS: Dose-limiting toxicities were hyperbilirubinemia and hepatic transaminase elevations for CI-treated patients in addition to mucositis and diarrhea for CIA-treated patients. MTD for CI was clofarabine 22.5 mg/m(2) intravenously daily x 5 and idarubicin 10 mg/m(2) intravenously daily x 3. MTD for CIA was clofarabine 22.5 mg/m(2) intravenously x 5, idarubicin 6 mg/m(2) intravenously x 3, and cytarabine 0.75 g/m(2) intravenously x 5 days.
CONCLUSIONS: A phase 2 randomized trial is in process to compare activity between treatment arms. (c) 2008 American Cancer Society.

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Year:  2008        PMID: 18756533      PMCID: PMC4163782          DOI: 10.1002/cncr.23816

Source DB:  PubMed          Journal:  Cancer        ISSN: 0008-543X            Impact factor:   6.860


  17 in total

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Journal:  Cancer Gene Ther       Date:  2003-01       Impact factor: 5.987

2.  Phase II study of clofarabine in pediatric patients with refractory or relapsed acute lymphoblastic leukemia.

Authors:  Sima Jeha; Paul S Gaynon; Bassem I Razzouk; Janet Franklin; Richard Kadota; Violet Shen; Lori Luchtman-Jones; Michael Rytting; Lisa R Bomgaars; Susan Rheingold; Kim Ritchey; Edythe Albano; Robert J Arceci; Stewart Goldman; Timothy Griffin; Arnold Altman; Bruce Gordon; Laurel Steinherz; Steven Weitman; Peter Steinherz
Journal:  J Clin Oncol       Date:  2006-04-20       Impact factor: 44.544

3.  Biochemical modulation of cytarabine triphosphate by clofarabine.

Authors:  Todd Cooper; Mary Ayres; Billie Nowak; Varsha Gandhi
Journal:  Cancer Chemother Pharmacol       Date:  2004-10-16       Impact factor: 3.333

4.  Preclinical antitumor activity of 2-chloro-9-(2-deoxy-2-fluoro-beta-D- arabinofuranosyl)adenine (Cl-F-ara-A).

Authors:  W R Waud; S M Schmid; J A Montgomery; J A Secrist
Journal:  Nucleosides Nucleotides Nucleic Acids       Date:  2000 Jan-Feb       Impact factor: 1.381

Review 5.  The treatment of acute myeloid leukemia in first relapse: a comprehensive review of the literature.

Authors:  Lance H Leopold; Roel Willemze
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6.  Results of a phase 1-2 study of clofarabine in combination with cytarabine (ara-C) in relapsed and refractory acute leukemias.

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7.  Synthesis and biologic activity of 2'-fluoro-2-halo derivatives of 9-beta-D-arabinofuranosyladenine.

Authors:  J A Montgomery; A T Shortnacy-Fowler; S D Clayton; J M Riordan; J A Secrist
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Review 8.  New agents in acute myeloid leukemia and other myeloid disorders.

Authors:  Farhad Ravandi; Hagop Kantarjian; Francis Giles; Jorge Cortes
Journal:  Cancer       Date:  2004-02-01       Impact factor: 6.860

9.  Phase I clinical and pharmacology study of clofarabine in patients with solid and hematologic cancers.

Authors:  Hagop M Kantarjian; Varsha Gandhi; Peter Kozuch; Stefan Faderl; Francis Giles; Jorge Cortes; Susan O'Brien; Nuhad Ibrahim; Fadlo Khuri; Min Du; Mary Beth Rios; Sima Jeha; Peter McLaughlin; William Plunkett; Michael Keating
Journal:  J Clin Oncol       Date:  2003-03-15       Impact factor: 44.544

10.  Phase 2 clinical and pharmacologic study of clofarabine in patients with refractory or relapsed acute leukemia.

Authors:  Hagop Kantarjian; Varsha Gandhi; Jorge Cortes; Srdan Verstovsek; Min Du; Guillermo Garcia-Manero; Francis Giles; Stefan Faderl; Susan O'Brien; Sima Jeha; Jan Davis; Zeev Shaked; Adam Craig; Michael Keating; William Plunkett; Emil J Freireich
Journal:  Blood       Date:  2003-06-05       Impact factor: 22.113

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  20 in total

1.  Report of a phase II study of clofarabine and cytarabine in de novo and relapsed and refractory AML patients and in selected elderly patients at high risk for anthracycline toxicity.

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Journal:  Oncologist       Date:  2011-01-27

2.  Phase 1 dose-escalation trial of clofarabine followed by escalating dose of fractionated cyclophosphamide in adults with relapsed or refractory acute leukaemias.

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Journal:  Br J Haematol       Date:  2012-05-18       Impact factor: 6.998

Review 3.  Interstrand crosslink inducing agents in pretransplant conditioning therapy for hematologic malignancies.

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Review 4.  Allogeneic hematopoietic cell transplantation in patients with AML not achieving remission: potentially curative therapy.

Authors:  B Gyurkocza; H M Lazarus; S Giralt
Journal:  Bone Marrow Transplant       Date:  2017-02-27       Impact factor: 5.483

5.  Prognostic implications of chromosome 17 abnormalities in the context of monosomal karyotype in patients with acute myeloid leukemia and complex cytogenetics.

Authors:  Aziz Nazha; Hagop M Kantarjian; Vijaya R Bhatt; Graciela Nogueras-Gonzalez; Jorge E Cortes; Tapan Kadia; Guillermo Garcia-Manero; Lynne Abruzzo; Naval Daver; Naveen Pemmaraju; Alfonso Quintas-Cardama; Farhad Ravandi; Michael Keating; Gautam Borthakur
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6.  Clofarabine in the treatment of acute myeloid leukemia in older adults.

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7.  Use of clofarabine for acute childhood leukemia.

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8.  Clofarabine, idarubicin, and cytarabine (CIA) as frontline therapy for patients ≤60 years with newly diagnosed acute myeloid leukemia.

Authors:  Aziz Nazha; Hagop Kantarjian; Farhad Ravandi; Xuelin Huang; Sangbum Choi; Guillermo Garcia-Manero; Elias Jabbour; Gautam Borthakur; Tapan Kadia; Marina Konopleva; Jorge Cortes; Alessandra Ferrajoli; Steve Kornblau; Naval Daver; Naveen Pemmaraju; Michael Andreeff; Zeev Estrov; Min Du; Mark Brandt; Stefan Faderl
Journal:  Am J Hematol       Date:  2013-09-09       Impact factor: 10.047

9.  Salvage therapy for relapsed or refractory acute myeloid leukemia.

Authors:  James K Mangan; Selina M Luger
Journal:  Ther Adv Hematol       Date:  2011-04

10.  A multicenter trial of myeloablative clofarabine and busulfan conditioning for relapsed or primary induction failure AML not in remission at the time of allogeneic hematopoietic stem cell transplantation.

Authors:  J Magenau; P Westervelt; S Khaled; J McGuirk; P Hari; M Eapen; P S Becker; B Parkin; T Braun; B Logan; H Wang; M Jagasia; S D Rowley; D D H Kim; T Schechter; N Frey; B Scott; T Churay; S Lieland; S Forman; S Mineishi
Journal:  Bone Marrow Transplant       Date:  2016-07-18       Impact factor: 5.483

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